| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA2153595 | 7e | PPB | 99.92 | % | ALA3301365 | % | |||||
| 2. | ALA2153595 | 7e | PPB | 99.57 | % | ALA3301368 | % | |||||
| 3. | ALA2153595 | 7e | CLint | 24.55 | microL/min/1E6 cells | ALA3301372 | uL.min-1.(10^6cells)-1 | |||||
| 4. | ALA2153595 | 7e | F | = | 87 | % | ALA2155517 | % | Rattus norvegicus | |||
| 5. | ALA2153595 | 7e | beta t1/2 | = | 3.4 | hr | ALA2155516 | hr | Rattus norvegicus | |||
| 6. | ALA2153595 | 7e | AUC | = | 471.5 | uM.hr | ALA2155515 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
| 7. | ALA2153595 | 7e | Cp | = | 40.5 | uM | ALA2155514 | uM | Rattus norvegicus | |||
| 8. | ALA2153595 | 7e | Cp | = | 70 | uM | ALA2155513 | uM | Rattus norvegicus | |||
| 9. | ALA2153595 | 7e | Tmax | = | 1.5 | hr | ALA2155512 | hr | Rattus norvegicus | |||
| 10. | ALA2153595 | 7e | Cmax | = | 72 | uM | ALA2155511 | nM | Rattus norvegicus | |||
| 11. | ALA2153595 | 7e | beta t1/2 | = | 1.3 | hr | ALA2155428 | hr | Rattus norvegicus | |||
| 12. | ALA2153595 | 7e | Vdss | = | 0.2 | L/Kg | ALA2155427 | L.kg-1 | Rattus norvegicus | |||
| 13. | ALA2153595 | 7e | CL | = | 2 | ml/min.kg | ALA2155426 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 14. | ALA2153595 | 7e | Cmax | = | 56 | uM | ALA2155425 | nM | Rattus norvegicus | |||
| 15. | ALA2153595 | 7e | IC50 | > | 20 | uM | ALA2155424 | nM | Homo sapiens | |||
| 16. | ALA2153595 | 7e | CLH | = | 0.17 | nmol/min/mg | ALA2155421 | nmol/min/mg | Rattus norvegicus | |||
| 17. | ALA2153595 | 7e | IC50 | = | 180 | nM | ALA2156127 | 6.75 | nM | Homo sapiens |
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