# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2153596 | 7f | Cp | = | 15 | uM | ALA2155434 | uM | Rattus norvegicus | |||
2. | ALA2153596 | 7f | Cp | = | 20 | uM | ALA2155433 | uM | Rattus norvegicus | |||
3. | ALA2153596 | 7f | Cp | = | 19 | uM | ALA2155432 | uM | Rattus norvegicus | |||
4. | ALA2153596 | 7f | AUC | = | 304 | uM.hr | ALA2155431 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
5. | ALA2153596 | 7f | Tmax | = | 2.7 | hr | ALA2155430 | hr | Rattus norvegicus | |||
6. | ALA2153596 | 7f | Cmax | = | 21 | uM | ALA2155429 | nM | Rattus norvegicus | |||
7. | ALA2153596 | 7f | beta t1/2 | = | 0.3 | hr | ALA2155428 | hr | Rattus norvegicus | |||
8. | ALA2153596 | 7f | Vdss | = | 0.1 | L/Kg | ALA2155427 | L.kg-1 | Rattus norvegicus | |||
9. | ALA2153596 | 7f | CL | = | 4.8 | ml/min.kg | ALA2155426 | mL.min-1.kg-1 | Rattus norvegicus | |||
10. | ALA2153596 | 7f | Cmax | = | 92 | uM | ALA2155425 | nM | Rattus norvegicus | |||
11. | ALA2153596 | 7f | IC50 | > | 30 | uM | ALA2155424 | nM | Homo sapiens | |||
12. | ALA2153596 | 7f | IC50 | = | 435 | nM | ALA2155423 | 6.36 | nM | Rattus norvegicus | ||
13. | ALA2153596 | 7f | CLH | = | 0.3 | nmol/min/mg | ALA2155421 | nmol/min/mg | Rattus norvegicus | |||
14. | ALA2153596 | 7f | IC50 | = | 160 | nM | ALA2156127 | 6.80 | nM | Homo sapiens |