# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2158561 | 36q | Ki | < | 1 | nM | ALA2162319 | nM | Homo sapiens | |||
2. | ALA2158561 | 36q | IC50 | > | 30 | uM | ALA2162322 | nM | Homo sapiens | |||
3. | ALA2158561 | 36q | IC50 | > | 30 | uM | ALA2162323 | nM | Homo sapiens | |||
4. | ALA2158561 | 36q | GI50 | = | 20 | nM | ALA2162324 | nM | Homo sapiens | |||
5. | ALA2158561 | 36q | GI50 | = | 131 | nM | ALA2162325 | nM | Homo sapiens | |||
6. | ALA2158561 | 36q | GI50 | = | 23 | nM | ALA2162326 | nM | Homo sapiens | |||
7. | ALA2158561 | 36q | Cmax | = | 11 | ng/ml | ALA2162329 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Mus musculus | ||
8. | ALA2158561 | 36q | Tmax | = | 0.25 | hr | ALA2162330 | hr | Mus musculus | |||
9. | ALA2158561 | 36q | Tmax | = | 0.5 | hr | ALA2162339 | hr | Mus musculus | |||
10. | ALA2158561 | 36q | Ratio | = | 2.6 | ALA2162340 | ||||||
11. | ALA2158561 | 36q | INH | 0 | ALA2162341 | Active | % | Homo sapiens | ||||
12. | ALA2158561 | 36q | INH | 0 | ALA2162342 | Active | % | Homo sapiens | ||||
13. | ALA2158561 | 36q | INH | 0 | ALA2162343 | Active | % | Homo sapiens | ||||
14. | ALA2158561 | 36q | INH | 0 | ALA2162498 | Active | % | Homo sapiens | ||||
15. | ALA2158561 | 36q | INH | 0 | ALA2162499 | Active | % | Homo sapiens | ||||
16. | ALA2158561 | 36q | AUC | = | 16 | ng/mL.hr | ALA2162502 | ng.hr.mL-1 | Mus musculus | |||
17. | ALA2158561 | 36q | AUC | = | 41 | ng/mL.hr | ALA2162503 | ng.hr.mL-1 | Mus musculus | |||
18. | ALA2158561 | 36q | CLH | = | 73 | microL/min/mg | ALA2162501 | mL.min-1.g-1 | Homo sapiens | |||
19. | ALA2158561 | 36q | ERH | = | 0.8 | ALA2162500 | Homo sapiens | |||||
20. | ALA2158561 | 36q | Cmax | = | 0.025 | uM | ALA2162329 | nM | Mus musculus |