| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA2158562 | 36r | Ki | < | 1 | nM | ALA2162319 | nM | Homo sapiens | |||
| 2. | ALA2158562 | 36r | Kd | = | 0.4 | nM | ALA2162320 | 9.40 | nM | |||
| 3. | ALA2158562 | 36r | Kd | < | 3 | nM | ALA2162321 | nM | ||||
| 4. | ALA2158562 | 36r | IC50 | > | 30 | uM | ALA2162322 | nM | Homo sapiens | |||
| 5. | ALA2158562 | 36r | IC50 | > | 30 | uM | ALA2162323 | nM | Homo sapiens | |||
| 6. | ALA2158562 | 36r | GI50 | = | 34 | nM | ALA2162324 | nM | Homo sapiens | |||
| 7. | ALA2158562 | 36r | GI50 | = | 32 | nM | ALA2162325 | nM | Homo sapiens | |||
| 8. | ALA2158562 | 36r | GI50 | = | 30 | nM | ALA2162326 | nM | Homo sapiens | |||
| 9. | ALA2158562 | 36r | AUC | = | 297 | ng/mL.hr | ALA2162327 | ng.hr.mL-1 | Mus musculus | |||
| 10. | ALA2158562 | 36r | t1/2 | = | 1.4 | hr | ALA2162328 | hr | Mus musculus | |||
| 11. | ALA2158562 | 36r | Cmax | = | 239 | ng/ml | ALA2162329 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Mus musculus | ||
| 12. | ALA2158562 | 36r | Tmax | = | 0.25 | hr | ALA2162330 | hr | Mus musculus | |||
| 13. | ALA2158562 | 36r | AUC | = | 231 | ng/mL.hr | ALA2162331 | ng.hr.mL-1 | Mus musculus | |||
| 14. | ALA2158562 | 36r | t1/2 | = | 2.4 | hr | ALA2162332 | hr | Mus musculus | |||
| 15. | ALA2158562 | 36r | Cmax | = | 68 | ng/ml | ALA2162333 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Mus musculus | ||
| 16. | ALA2158562 | 36r | Tmax | = | 0.25 | hr | ALA2162334 | hr | Mus musculus | |||
| 17. | ALA2158562 | 36r | Ratio | = | 0.8 | ALA2162335 | ||||||
| 18. | ALA2158562 | 36r | AUC | = | 6915 | ng/mL.hr | ALA2162336 | ng.hr.mL-1 | Mus musculus | |||
| 19. | ALA2158562 | 36r | t1/2 | = | 1.2 | hr | ALA2162337 | hr | Mus musculus | |||
| 20. | ALA2158562 | 36r | Cmax | = | 5389 | ng/ml | ALA2162338 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Mus musculus |
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