# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2159536 | 27 | deltaTm | = | 7.9 | degrees C | ALA2161770 | degrees C | ||||
2. | ALA2159536 | 27 | Ratio EC50 | = | 147 | ALA2162452 | ||||||
3. | ALA2159536 | 27 | Ratio EC50 | = | 147 | ALA2162453 | ||||||
4. | ALA2159536 | 27 | IC50 | = | 19 | nM | ALA2161885 | 7.72 | nM | |||
5. | ALA2159536 | 27 | IC50 | = | 6591 | nM | ALA2161886 | 5.18 | nM | Homo sapiens | ||
6. | ALA2159536 | 27 | Ratio IC50 | = | 347 | ALA2161887 | ||||||
7. | ALA2159536 | 27 | EC50 | = | 150 | nM | ALA2161888 | 6.82 | nM | Trypanosoma brucei brucei | ||
8. | ALA2159536 | 27 | EC50 | = | 22000 | nM | ALA2161889 | 4.66 | nM | |||
9. | ALA2159536 | 27 | EC50 | = | 22000 | nM | ALA2161890 | 4.66 | nM | Homo sapiens | ||
10. | ALA2159536 | 27 | AQ | = | 0.53 | ALA2162449 | Homo sapiens | |||||
11. | ALA2159536 | 27 | Papp | = | 191 | nm/s | ALA2161891 | nm/s | ||||
12. | ALA2159536 | 27 | Papp | = | 97 | nm/s | ALA2161892 | nm/s | ||||
13. | ALA2159536 | 27 | Cmax | = | 1.29 | uM | ALA2161894 | nM | Mus musculus | |||
14. | ALA2159536 | 27 | Tmax | = | 30 | min | ALA2162442 | hr | Mus musculus | |||
15. | ALA2159536 | 27 | t1/2 | = | 82 | min | ALA2162443 | hr | Mus musculus | |||
16. | ALA2159536 | 27 | AUC | = | 161 | uM.min | ALA2162444 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Mus musculus |