# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2163360 | 39 | LogD7.4 | 2.13 | ALA3301363 | |||||||
2. | ALA2163360 | 39 | CLint | 7 | microL/min/mg | ALA3301370 | mL.min-1.g-1 | |||||
3. | ALA2163360 | 39 | CLint | < | 3 | microL/min/1E6 cells | ALA3301371 | uL.min-1.(10^6cells)-1 | ||||
4. | ALA2163360 | 39 | Solubility | 1513.6 | uM | ALA3301364 | nM | |||||
5. | ALA2163360 | 39 | IC50 | = | 0.001 | uM | ALA2168708 | 9.00 | nM | Homo sapiens | ||
6. | ALA2163360 | 39 | IC50 | 0 | ALA2168709 | Not Active | Homo sapiens | |||||
7. | ALA2163360 | 39 | IC50 | > | 4 | uM | ALA2168710 | nM | Homo sapiens | |||
8. | ALA2163360 | 39 | IC50 | > | 2.9 | uM | ALA2168711 | nM | Homo sapiens | |||
9. | ALA2163360 | 39 | logD | = | 2.1 | ALA2168713 | ||||||
10. | ALA2163360 | 39 | solubility | = | 1500 | uM | ALA2168929 | nM | ||||
11. | ALA2163360 | 39 | CLH | = | 12 | microL/min/mg | ALA2168927 | mL.min-1.g-1 | Homo sapiens | |||
12. | ALA2163360 | 39 | CLH | = | 25 | microL/min/mg | ALA2168931 | mL.min-1.g-1 | Rattus norvegicus | |||
13. | ALA2163360 | 39 | Fu | = | 42 | % | ALA2168930 | Rattus norvegicus | ||||
14. | ALA2163360 | 39 | Fu | = | 38 | % | ALA2168928 | Canis lupus familiaris | ||||
15. | ALA2163360 | 39 | CLH | = | 3.1 | uL/min | ALA2168714 | uL/min | ||||
16. | ALA2163360 | 39 | CL | = | 32 | ml/min.kg | ALA2168715 | mL.min-1.kg-1 | Rattus norvegicus | |||
17. | ALA2163360 | 39 | CL | = | 7.2 | ml/min.kg | ALA2168716 | mL.min-1.kg-1 | Canis lupus familiaris | |||
18. | ALA2163360 | 39 | Vdss | = | 1.6 | L/Kg | ALA2168717 | L.kg-1 | Rattus norvegicus | |||
19. | ALA2163360 | 39 | Vdss | = | 0.9 | L/Kg | ALA2168917 | L.kg-1 | Canis lupus familiaris | |||
20. | ALA2163360 | 39 | t1/2 | = | 1.8 | hr | ALA2168918 | hr | Rattus norvegicus |