# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2165084 | 5d | Retention_time | = | 13.72 | min | ALA4409103 | min | ||||
2. | ALA2165084 | 5d | Activity | 0 | ALA4409102 | Active | Homo sapiens | |||||
3. | ALA2165084 | 5d | Activity | 0 | ALA4409101 | Active | Homo sapiens | |||||
4. | ALA2165084 | 5d | Activity | 0 | ALA4409100 | Non-Toxic | Homo sapiens | |||||
5. | ALA2165084 | 5d | t1/2 | = | 27.77 | min | ALA4409099 | hr | ||||
6. | ALA2165084 | 5d | CLH | = | 41.6 | microL/min/mg | ALA4409098 | mL.min-1.g-1 | ||||
7. | ALA2165084 | 5d | K | = | 0.025 | 10'-1/min | ALA4409097 | 10'-1/min | ||||
8. | ALA2165084 | 5d | t1/2 | = | 50.26 | min | ALA4409096 | hr | ||||
9. | ALA2165084 | 5d | CLH | = | 23.45 | microL/min/mg | ALA4409095 | mL.min-1.g-1 | ||||
10. | ALA2165084 | 5d | K | = | 0.014 | 10'-1/min | ALA4409094 | 10'-1/min | ||||
11. | ALA2165084 | 5d | IC50 | = | 50 | uM | ALA4409089 | 4.30 | nM | Homo sapiens | ||
12. | ALA2165084 | 5d | IC50 | = | 75 | uM | ALA4409088 | 4.12 | nM | Mus musculus | ||
13. | ALA2165084 | 5d | Stability | = | 92.1 | % | ALA4409087 | % | ||||
14. | ALA2165084 | 5d | solubility | 0 | ALA4409086 | Bld | ||||||
15. | ALA2165084 | 5d | solubility | = | 465 | uM | ALA4409085 | nM | ||||
16. | ALA2165084 | 5d | Ki | = | 0.16 | nM | ALA2168075 | 9.80 | nM | Mus musculus | ||
17. | ALA2165084 | 5d | IC50 | = | 0.6 | nM | ALA2168075 | 9.22 | nM | Mus musculus | ||
18. | ALA2165084 | 5d | IC50 | 0 | ALA2168070 | Not Determined | Homo sapiens | |||||
19. | ALA2165084 | 5d | INH | 0 | ALA2168069 | Active | % | Mus musculus | ||||
20. | ALA2165084 | 5d | INH | 0 | ALA2167888 | Active | % | Mus musculus |