# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2170835 | 28 | IC50 | = | 10.2 | nM | ALA2173962 | 7.99 | nM | Homo sapiens | ||
2. | ALA2170835 | 28 | Ki | = | 2.4 | nM | ALA2173961 | 8.62 | nM | Homo sapiens | ||
3. | ALA2170835 | 28 | IC50 | = | 7 | nM | ALA2173960 | 8.15 | nM | |||
4. | ALA2170835 | 28 | Ki | < | 1 | nM | ALA2173959 | nM | ||||
5. | ALA2170835 | 28 | Activity | 0 | ALA2173958 | Not Active | Homo sapiens | |||||
6. | ALA2170835 | 28 | IC50 | = | 125 | nM | ALA2173957 | 6.90 | nM | Homo sapiens | ||
7. | ALA2170835 | 28 | IC50 | = | 108 | nM | ALA2173956 | 6.97 | nM | |||
8. | ALA2170835 | 28 | Activity | 0 | ALA2173955 | Dose-dependent effect | Homo sapiens | |||||
9. | ALA2170835 | 28 | MTD | = | 50 | mg kg-1 | ALA2173950 | mg kg-1 | Mus musculus | |||
10. | ALA2170835 | 28 | Activity | < | 10 | % | ALA2173947 | % | Mus musculus | |||
11. | ALA2170835 | 28 | Activity | > | 10 | % | ALA2173871 | % | Mus musculus | |||
12. | ALA2170835 | 28 | TGI | 0 | ALA2173868 | Active | ||||||
13. | ALA2170835 | 28 | Activity | 0 | ALA2173867 | Not Active | ||||||
14. | ALA2170835 | 28 | Activity | 0 | ALA2173864 | Active | Homo sapiens | |||||
15. | ALA2170835 | 28 | Activity | 0 | ALA2173863 | Active | Homo sapiens | |||||
16. | ALA2170835 | 28 | Activity | 0 | ALA2173860 | Active | Homo sapiens | |||||
17. | ALA2170835 | 28 | Activity | 0 | ALA2173859 | Active | Homo sapiens |