# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2171421 | 7 | IC50 | = | 31 | nM | ALA2174779 | 7.51 | nM | Homo sapiens | ||
2. | ALA2171421 | 7 | IC50 | = | 6.55 | uM | ALA2174683 | 5.18 | nM | Homo sapiens | ||
3. | ALA2171421 | 7 | IC50 | = | 43 | nM | ALA2174777 | 7.37 | nM | Homo sapiens | ||
4. | ALA2171421 | 7 | INH | = | 37 | % | ALA2174776 | % | Homo sapiens | |||
5. | ALA2171421 | 7 | INH | = | 29 | % | ALA2174775 | % | Homo sapiens | |||
6. | ALA2171421 | 7 | INH | = | 6 | % | ALA2174774 | % | Homo sapiens | |||
7. | ALA2171421 | 7 | INH | = | 86 | % | ALA2174773 | % | Homo sapiens | |||
8. | ALA2171421 | 7 | INH | = | 3 | % | ALA2174772 | % | Homo sapiens | |||
9. | ALA2171421 | 7 | INH | = | 0 | % | ALA2174771 | % | Homo sapiens | |||
10. | ALA2171421 | 7 | INH | = | 9 | % | ALA2174770 | % | Homo sapiens | |||
11. | ALA2171421 | 7 | INH | = | 23 | % | ALA2174769 | % | Homo sapiens | |||
12. | ALA2171421 | 7 | INH | = | 10 | % | ALA2174768 | % | Homo sapiens | |||
13. | ALA2171421 | 7 | Ratio IC50 | > | 200 | ALA2174682 | ||||||
14. | ALA2171421 | 7 | Ratio IC50 | > | 150 | ALA2174680 | ||||||
15. | ALA2171421 | 7 | Stability | = | 43 | % | ALA2174681 | % | Homo sapiens | |||
16. | ALA2171421 | 7 | Stability | = | 68 | % | ALA2174679 | % | Rattus norvegicus | |||
17. | ALA2171421 | 7 | Stability | = | 4 | % | ALA2174678 | % | Mus musculus | |||
18. | ALA2171421 | 7 | Drug uptake | = | 1138 | ng/g | ALA2174677 | ng/g | Mus musculus | |||
19. | ALA2171421 | 7 | Cp | = | 699 | ng/ml | ALA2174676 | ng/ml | Mus musculus | |||
20. | ALA2171421 | 7 | BPR | = | 1.69 | ALA2174674 |