# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2171700 | 2c, MpPPOX | IC50 | = | 78 | nM | ALA4765584 | 7.11 | nM | Homo sapiens | ||
2. | ALA2171700 | 2c, MpPPOX | XI50 | > | 400 | molar excess | ALA4718660 | molar excess | Homo sapiens | |||
3. | ALA2171700 | 2c, MpPPOX | INH | = | 4 | % | ALA4718659 | % | Homo sapiens | |||
4. | ALA2171700 | 2c, MpPPOX | XI50 | > | 400 | molar excess | ALA4718658 | molar excess | Sus scrofa | |||
5. | ALA2171700 | 2c, MpPPOX | INH | = | 34.1 | % | ALA4718657 | % | Sus scrofa | |||
6. | ALA2171700 | 2c, MpPPOX | IC50 | = | 31 | nM | ALA4202162 | 7.51 | nM | Homo sapiens | ||
7. | ALA2171700 | 2c, MpPPOX | INH | 0 | ALA4202165 | Tde | % | Homo sapiens | ||||
8. | ALA2171700 | 2c, MpPPOX | IC50 | = | 1700 | nM | ALA4202164 | 5.77 | nM | Homo sapiens | ||
9. | ALA2171700 | 2c, MpPPOX | IC50 | = | 6.1 | nM | ALA3223064 | 8.21 | nM | Homo sapiens | ||
10. | ALA2171700 | 2c, MpPPOX | IC50 | = | 0.31 | uM | ALA2379576 | 6.51 | nM | Homo sapiens | ||
11. | ALA2171700 | 2c, MpPPOX | IC50 | = | 0.72 | uM | ALA2379575 | 6.14 | nM | Rattus norvegicus | ||
12. | ALA2171700 | 2c, MpPPOX | IC50 | = | 0.078 | uM | ALA2379563 | 7.11 | nM | Homo sapiens | ||
13. | ALA2171700 | 2c, MpPPOX | IC50 | = | 0.065 | uM | ALA2379560 | 7.19 | nM | Homo sapiens | ||
14. | ALA2171700 | 2c, MpPPOX | XI50 | > | 400 | molar excess | ALA2174474 | molar excess | Homo sapiens | |||
15. | ALA2171700 | 2c, MpPPOX | XI50 | = | 57.6 | molar excess | ALA2174473 | molar excess | Sus scrofa | |||
16. | ALA2171700 | 2c, MpPPOX | XI50 | = | 1.04 | molar excess | ALA2174472 | molar excess | Homo sapiens | |||
17. | ALA2171700 | 2c, MpPPOX | XI50 | > | 40 | molar excess | ALA2174470 | molar excess | Cavia porcellus | |||
18. | ALA2171700 | 2c, MpPPOX | XI50 | = | 7.12 | molar excess | ALA2174469 | molar excess | Canis familiaris | |||
19. | ALA2171700 | 2c, MpPPOX | XI50 | = | 0.93 | molar excess | ALA2174471 | molar excess | Homo sapiens | |||
20. | ALA2171700 | 2c, MpPPOX | t1/2 | > | 120 | min | ALA2174468 | hr | Homo sapiens |