# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2177539 | (+)-12a | Ki | = | 9.4 | nM | ALA2187477 | 8.03 | nM | Homo sapiens | ||
2. | ALA2177539 | (+)-12a | Ki | = | 70 | nM | ALA2187476 | 7.16 | nM | Homo sapiens | ||
3. | ALA2177539 | (+)-12a | Ki | = | 1796 | nM | ALA2187475 | 5.75 | nM | Homo sapiens | ||
4. | ALA2177539 | (+)-12a | %max | = | 53 | % | ALA2187471 | % | Homo sapiens | |||
5. | ALA2177539 | (+)-12a | EC50 | = | 6661 | nM | ALA2187470 | 5.18 | nM | Homo sapiens | ||
6. | ALA2177539 | (+)-12a | %max | = | 17 | % | ALA2187469 | % | Homo sapiens | |||
7. | ALA2177539 | (+)-12a | EC50 | > | 10000 | nM | ALA2187468 | nM | Homo sapiens | |||
8. | ALA2177539 | (+)-12a | %max | = | 25 | % | ALA2187467 | % | Homo sapiens | |||
9. | ALA2177539 | (+)-12a | EC50 | > | 10000 | nM | ALA2187466 | nM | Homo sapiens | |||
10. | ALA2177539 | (+)-12a | %max | = | 18 | % | ALA2187465 | % | Homo sapiens | |||
11. | ALA2177539 | (+)-12a | EC50 | = | 3.1 | uM | ALA2187464 | 5.51 | nM | Homo sapiens | ||
12. | ALA2177539 | (+)-12a | %max | = | 87 | % | ALA2187463 | % | ||||
13. | ALA2177539 | (+)-12a | EC50 | = | 6 | uM | ALA2187462 | 5.22 | nM | |||
14. | ALA2177539 | (+)-12a | %max | = | 13 | % | ALA2187461 | % | Rattus norvegicus | |||
15. | ALA2177539 | (+)-12a | EC50 | = | 855 | nM | ALA2187459 | 6.07 | nM | Rattus norvegicus | ||
16. | ALA2177539 | (+)-12a | Ki | = | 320 | nM | ALA2187460 | 6.50 | nM | Homo sapiens | ||
17. | ALA2177539 | (+)-12a | %max | = | 9 | % | ALA2187043 | % | ||||
18. | ALA2177539 | (+)-12a | EC50 | > | 10000 | nM | ALA2185176 | nM |