# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2178135 | 19 | Ki | = | 1 | nM | ALA2188383 | 9.00 | nM | Homo sapiens | ||
2. | ALA2178135 | 19 | Ratio Ki | > | 3200 | ALA2188380 | ||||||
3. | ALA2178135 | 19 | IC50 | = | 4 | nM | ALA2188381 | 8.40 | nM | Homo sapiens | ||
4. | ALA2178135 | 19 | CLH | = | 4.9 | ml/min.kg | ALA2188378 | mL.min-1.kg-1 | Homo sapiens | |||
5. | ALA2178135 | 19 | CLH | = | 15 | ml/min.kg | ALA2188377 | mL.min-1.kg-1 | Rattus norvegicus | |||
6. | ALA2178135 | 19 | PPB | = | 97.6 | % | ALA2188376 | % | Rattus norvegicus | |||
7. | ALA2178135 | 19 | Papp | = | 10.9 | ucm/s | ALA2188375 | ucm/s | Canis lupus familiaris | |||
8. | ALA2178135 | 19 | Ratio | = | 1.3 | ALA2188374 | Canis lupus familiaris | |||||
9. | ALA2178135 | 19 | Ratio Ki | = | 118 | ALA2188369 | ||||||
10. | ALA2178135 | 19 | INH | > | 70 | % | ALA2188363 | % | Homo sapiens | |||
11. | ALA2178135 | 19 | INH | 0 | ALA2187978 | Active | % | Mus musculus | ||||
12. | ALA2178135 | 19 | INH | 0 | ALA2187977 | Active | % | Mus musculus | ||||
13. | ALA2178135 | 19 | CLH | = | 9.2 | ml/min.kg | ALA2187976 | mL.min-1.kg-1 | ||||
14. | ALA2178135 | 19 | PPB | = | 95.5 | % | ALA2187975 | % | Macaca fascicularis |