# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2179435 | Ac-LLLLRVKR-NH2 | IC50 | = | 30 | nM | ALA5151873 | 7.52 | nM | Homo sapiens | ||
2. | ALA2179435 | Ac-LLLLRVKR-NH2 | IC50 | = | 20 | nM | ALA5151867 | 7.70 | nM | Homo sapiens | ||
3. | ALA2179435 | Ac-LLLLRVKR-NH2 | IC50 | = | 25 | uM | ALA4261464 | 4.60 | nM | Homo sapiens | ||
4. | ALA2179435 | Ac-LLLLRVKR-NH2 | IC50 | = | 45 | uM | ALA4261465 | 4.35 | nM | Homo sapiens | ||
5. | ALA2179435 | Ac-LLLLRVKR-NH2 | t1/2 | = | 1.7 | hr | ALA4261467 | hr | ||||
6. | ALA2179435 | Ac-LLLLRVKR-NH2 | IC50 | = | 100 | uM | ALA4236736 | 4.00 | nM | Homo sapiens | ||
7. | ALA2179435 | Ac-LLLLRVKR-NH2 | IC50 | = | 180 | uM | ALA4236737 | nM | Homo sapiens | |||
8. | ALA2179435 | Ac-LLLLRVKR-NH2 | Ratio Ki | = | 20 | ALA4236738 | ||||||
9. | ALA2179435 | Ac-LLLLRVKR-NH2 | Ki | = | 430 | nM | ALA4236739 | 6.37 | nM | Homo sapiens | ||
10. | ALA2179435 | Ac-LLLLRVKR-NH2 | Ki | = | 22 | nM | ALA4236727 | 7.66 | nM | Homo sapiens | ||
11. | ALA2179435 | Ac-LLLLRVKR-NH2 | Ki | = | 20 | nM | ALA3117754 | 7.70 | nM | Homo sapiens | ||
12. | ALA2179435 | Ac-LLLLRVKR-NH2 | Ki | = | 430 | nM | ALA3117753 | 6.37 | nM | Homo sapiens | ||
13. | ALA2179435 | Ac-LLLLRVKR-NH2 | Stability | 0 | ALA3117755 | Unstable | % | Mus musculus | ||||
14. | ALA2179435 | Ac-LLLLRVKR-NH2 | IC50 | = | 100 | uM | ALA3117748 | 4.00 | nM | Homo sapiens | ||
15. | ALA2179435 | Ac-LLLLRVKR-NH2 | INH | < | 50 | % | ALA3117743 | % | Homo sapiens | |||
16. | ALA2179435 | Ac-LLLLRVKR-NH2 | INH | < | 5 | % | ALA3117742 | % | Homo sapiens | |||
17. | ALA2179435 | Ac-LLLLRVKR-NH2 | Drug uptake | 0 | ALA3117741 | Active | Homo sapiens | |||||
18. | ALA2179435 | Ac-LLLLRVKR-NH2 | t1/2 | = | 5.1 | hr | ALA3117749 | hr | Mus musculus | |||
19. | ALA2179435 | Ac-LLLLRVKR-NH2 | IC50 | = | 180 | uM | ALA3117746 | nM | Homo sapiens | |||
20. | ALA2179435 | Ac-LLLLRVKR-NH2 | Activity | = | 1 | % | ALA2187686 | % | Homo sapiens |