# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2179834 | Ac-[DLeu]LLLRVKR-NH2 | Ki | = | 24 | nM | ALA4261461 | 7.62 | nM | Homo sapiens | ||
2. | ALA2179834 | Ac-[DLeu]LLLRVKR-NH2 | Ki | = | 760 | nM | ALA4261462 | 6.12 | nM | Homo sapiens | ||
3. | ALA2179834 | Ac-[DLeu]LLLRVKR-NH2 | Ratio Ki | = | 32 | ALA4261463 | ||||||
4. | ALA2179834 | Ac-[DLeu]LLLRVKR-NH2 | IC50 | = | 70 | uM | ALA4261464 | 4.16 | nM | Homo sapiens | ||
5. | ALA2179834 | Ac-[DLeu]LLLRVKR-NH2 | IC50 | = | 150 | uM | ALA4261465 | nM | Homo sapiens | |||
6. | ALA2179834 | Ac-[DLeu]LLLRVKR-NH2 | Ki | = | 24 | nM | ALA3117754 | 7.62 | nM | Homo sapiens | ||
7. | ALA2179834 | Ac-[DLeu]LLLRVKR-NH2 | Ki | = | 760 | nM | ALA3117753 | 6.12 | nM | Homo sapiens | ||
8. | ALA2179834 | Ac-[DLeu]LLLRVKR-NH2 | Ratio Ki | <= | 32 | ALA3117752 | ||||||
9. | ALA2179834 | Ac-[DLeu]LLLRVKR-NH2 | t1/2 | = | 8.6 | hr | ALA3117749 | hr | Mus musculus | |||
10. | ALA2179834 | Ac-[DLeu]LLLRVKR-NH2 | Stability | 0 | ALA3117755 | Unstable | % | Mus musculus | ||||
11. | ALA2179834 | Ac-[DLeu]LLLRVKR-NH2 | IC50 | = | 70 | uM | ALA3117748 | 4.16 | nM | Homo sapiens | ||
12. | ALA2179834 | Ac-[DLeu]LLLRVKR-NH2 | IC50 | = | 150 | uM | ALA3117746 | nM | Homo sapiens | |||
13. | ALA2179834 | Ac-[DLeu]LLLRVKR-NH2 | INH | < | 5 | % | ALA3117742 | % | Homo sapiens | |||
14. | ALA2179834 | Ac-[DLeu]LLLRVKR-NH2 | Drug uptake | 0 | ALA3117741 | Active | Homo sapiens | |||||
15. | ALA2179834 | Ac-[DLeu]LLLRVKR-NH2 | IC50 | = | 190 | uM | ALA3117744 | nM | Homo sapiens | |||
16. | ALA2179834 | Ac-[DLeu]LLLRVKR-NH2 | Activity | = | 0.4 | % | ALA2187686 | % | Homo sapiens | |||
17. | ALA2179834 | Ac-[DLeu]LLLRVKR-NH2 | Activity | = | 8.3 | % | ALA2187687 | % | Homo sapiens | |||
18. | ALA2179834 | Ac-[DLeu]LLLRVKR-NH2 | Activity | = | 8.4 | % | ALA2187689 | % | Homo sapiens | |||
19. | ALA2179834 | Ac-[DLeu]LLLRVKR-NH2 | Activity | = | 8.9 | % | ALA2187688 | % | Homo sapiens | |||
20. | ALA2179834 | Ac-[DLeu]LLLRVKR-NH2 | Activity | = | 11.8 | % | ALA2187690 | % | Homo sapiens |