# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2181202 | H-Dmt-D-Arg-Phe-Lys-NH2 | Ki | = | 877 | nM | ALA3783009 | 6.06 | nM | Rattus norvegicus | ||
2. | ALA2181202 | H-Dmt-D-Arg-Phe-Lys-NH2 | Ki | = | 0.58 | nM | ALA3783008 | 9.24 | nM | Rattus norvegicus | ||
3. | ALA2181202 | H-Dmt-D-Arg-Phe-Lys-NH2 | IC50 | = | 23.1 | nM | ALA3783007 | 7.64 | nM | Mus musculus | ||
4. | ALA2181202 | H-Dmt-D-Arg-Phe-Lys-NH2 | IC50 | = | 1.41 | nM | ALA3783006 | 8.85 | nM | Cavia porcellus | ||
5. | ALA2181202 | H-Dmt-D-Arg-Phe-Lys-NH2 | IC50 | = | 1.41 | nM | ALA3762578 | 8.85 | nM | Cavia porcellus | ||
6. | ALA2181202 | H-Dmt-D-Arg-Phe-Lys-NH2 | Ki | = | 2100 | nM | ALA3762573 | 5.68 | nM | Homo sapiens | ||
7. | ALA2181202 | H-Dmt-D-Arg-Phe-Lys-NH2 | Ki | = | 0.143 | nM | ALA3762577 | 9.85 | nM | Homo sapiens | ||
8. | ALA2181202 | H-Dmt-D-Arg-Phe-Lys-NH2 | ED50 | = | 6 | ug/kg | ALA5127602 | mg.kg-1 | ||||
9. | ALA2181202 | H-Dmt-D-Arg-Phe-Lys-NH2 | Ki | = | 2407 | nM | ALA5127592 | 5.62 | nM | Homo sapiens | ||
10. | ALA2181202 | H-Dmt-D-Arg-Phe-Lys-NH2 | Ki | = | 11.5 | nM | ALA5127591 | 7.94 | nM | Mus musculus | ||
11. | ALA2181202 | H-Dmt-D-Arg-Phe-Lys-NH2 | Ki | = | 115.7 | nM | ALA5127590 | 6.94 | nM | |||
12. | ALA2181202 | H-Dmt-D-Arg-Phe-Lys-NH2 | Ki | = | 0.14 | nM | ALA5127589 | 9.85 | nM | Bos taurus | ||
13. | ALA2181202 | H-Dmt-D-Arg-Phe-Lys-NH2 | ED50 | = | 22 | nmol | ALA5127581 | nmol | Mus musculus | |||
14. | ALA2181202 | H-Dmt-D-Arg-Phe-Lys-NH2 | ED50 | = | 1.1 | pmol | ALA5127570 | pmol | Mus musculus | |||
15. | ALA2181202 | H-Dmt-D-Arg-Phe-Lys-NH2 | ED50 | = | 61 | fmol | ALA5127570 | fmol | Mus musculus | |||
16. | ALA2181202 | H-Dmt-D-Arg-Phe-Lys-NH2 | IC50 | = | 23.1 | nM | ALA5127552 | 7.64 | nM | Mus musculus | ||
17. | ALA2181202 | H-Dmt-D-Arg-Phe-Lys-NH2 | IC50 | = | 1.41 | nM | ALA5127551 | 8.85 | nM | Cavia porcellus | ||
18. | ALA2181202 | H-Dmt-D-Arg-Phe-Lys-NH2 | ED50 | = | 65.5 | ug/kg | ALA5127511 | mg.kg-1 | Mus musculus | |||
19. | ALA2181202 | H-Dmt-D-Arg-Phe-Lys-NH2 | permeability | = | 3.64 | 10'-7nmol/cm2/min | ALA3269828 | 10'-7nmol/cm2/min | Homo sapiens | |||
20. | ALA2181202 | H-Dmt-D-Arg-Phe-Lys-NH2 | permeability | = | 3.13 | 10'-7nmol/cm2/min | ALA3269827 | 10'-7nmol/cm2/min | Homo sapiens |