# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2181202 | H-Dmt-D-Arg-Phe-Lys-NH2 | Ki | = | 0.143 | nM | ALA2182467 | 9.85 | nM | Homo sapiens | ||
2. | ALA2181202 | H-Dmt-D-Arg-Phe-Lys-NH2 | Ratio Ki | = | 7 | ALA2182465 | Homo sapiens | |||||
3. | ALA2181202 | H-Dmt-D-Arg-Phe-Lys-NH2 | t1/2 | = | 1.8 | hr | ALA2182466 | hr | Ovis aries | |||
4. | ALA2181202 | H-Dmt-D-Arg-Phe-Lys-NH2 | Ratio | = | 3000 | ALA2182464 | Rattus norvegicus | |||||
5. | ALA2181202 | H-Dmt-D-Arg-Phe-Lys-NH2 | Ki | = | 0.143 | nM | ALA2189109 | 9.85 | nM | Rattus norvegicus | ||
6. | ALA2181202 | H-Dmt-D-Arg-Phe-Lys-NH2 | Ki | = | 2100 | nM | ALA2189108 | 5.68 | nM | Rattus norvegicus | ||
7. | ALA2181202 | H-Dmt-D-Arg-Phe-Lys-NH2 | Ki | = | 22.3 | nM | ALA2189107 | 7.65 | nM | Cavia porcellus | ||
8. | ALA2181202 | H-Dmt-D-Arg-Phe-Lys-NH2 | Ratio Ki | = | 11400 | ALA2189106 | ||||||
9. | ALA2181202 | H-Dmt-D-Arg-Phe-Lys-NH2 | Ratio Ki | = | 156 | ALA2188652 | ||||||
10. | ALA2181202 | H-Dmt-D-Arg-Phe-Lys-NH2 | IC50 | = | 1.41 | nM | ALA2188651 | 8.85 | nM | Cavia porcellus | ||
11. | ALA2181202 | H-Dmt-D-Arg-Phe-Lys-NH2 | IC50 | = | 23.1 | nM | ALA2188650 | 7.64 | nM | Mus musculus | ||
12. | ALA2181202 | H-Dmt-D-Arg-Phe-Lys-NH2 | Kin | = | 9.44 | uL/g.min | ALA2188649 | uL/g.min | Mus musculus | |||
13. | ALA2181202 | H-Dmt-D-Arg-Phe-Lys-NH2 | Vz | = | 19.25 | uL/g | ALA2188648 | uL/g | Mus musculus | |||
14. | ALA2181202 | H-Dmt-D-Arg-Phe-Lys-NH2 | Drug uptake | = | 23.12 | % | ALA2188647 | % | Mus musculus | |||
15. | ALA2181202 | H-Dmt-D-Arg-Phe-Lys-NH2 | Drug uptake | = | 76.88 | % | ALA2188645 | % | Mus musculus | |||
16. | ALA2181202 | H-Dmt-D-Arg-Phe-Lys-NH2 | Activity | = | 0.058 | /min | ALA2188646 | /min | Mus musculus | |||
17. | ALA2181202 | H-Dmt-D-Arg-Phe-Lys-NH2 | Drug uptake | 0 | ALA2188643 | Active | Mus musculus | |||||
18. | ALA2181202 | H-Dmt-D-Arg-Phe-Lys-NH2 | Drug uptake | 0 | ALA2188642 | Active | Mus musculus | |||||
19. | ALA2181202 | H-Dmt-D-Arg-Phe-Lys-NH2 | Stability | = | 94.7 | % | ALA2188640 | % | Mus musculus | |||
20. | ALA2181202 | H-Dmt-D-Arg-Phe-Lys-NH2 | Stability | = | 102.6 | % | ALA2188641 | % | Mus musculus |