| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA2181928 | 8 | INH | = | 105 | % | ALA4423294 | % | Homo sapiens | |||
| 2. | ALA2181928 | 8 | pIC50 | = | 6.7 | ALA4423293 | 6.70 | nM | Homo sapiens | |||
| 3. | ALA2181928 | 8 | logD | = | 2.7 | ALA4423288 | ||||||
| 4. | ALA2181928 | 8 | pKi | = | 7.6 | ALA4423290 | 7.60 | nM | Homo sapiens | |||
| 5. | ALA2181928 | 8 | CLint | 52.48 | microL/min/1E6 cells | ALA3301371 | uL.min-1.(10^6cells)-1 | |||||
| 6. | ALA2181928 | 8 | PPB | 93.67 | % | ALA3301365 | % | |||||
| 7. | ALA2181928 | 8 | PPB | 90.72 | % | ALA3301366 | % | |||||
| 8. | ALA2181928 | 8 | LogD7.4 | 2.75 | ALA3301363 | |||||||
| 9. | ALA2181928 | 8 | CLint | 11.75 | microL/min/mg | ALA3301370 | mL.min-1.g-1 | |||||
| 10. | ALA2181928 | 8 | Ki | = | 6.3 | nM | ALA4028141 | 8.20 | nM | Homo sapiens | ||
| 11. | ALA2181928 | 8 | IC50 | = | 25 | nM | ALA4028141 | 7.60 | nM | Homo sapiens | ||
| 12. | ALA2181928 | 8 | IC50 | = | 44 | nM | ALA4028145 | 7.36 | nM | Homo sapiens | ||
| 13. | ALA2181928 | 8 | IC50 | > | 10000 | nM | ALA4028146 | nM | Homo sapiens | |||
| 14. | ALA2181928 | 8 | IC50 | > | 10000 | nM | ALA4028148 | nM | Homo sapiens | |||
| 15. | ALA2181928 | 8 | IC50 | > | 10000 | nM | ALA4028149 | nM | Homo sapiens | |||
| 16. | ALA2181928 | 8 | CLH | = | 287 | microL/min/mg | ALA4028152 | mL.min-1.g-1 | Rattus norvegicus | |||
| 17. | ALA2181928 | 8 | CLH | = | 6.9 | microL/min/mg | ALA4028150 | mL.min-1.g-1 | Homo sapiens | |||
| 18. | ALA2181928 | 8 | INH | < | 20 | % | ALA4028153 | % | Homo sapiens | |||
| 19. | ALA2181928 | 8 | INH | < | 20 | % | ALA4028154 | % | Homo sapiens | |||
| 20. | ALA2181928 | 8 | INH | < | 20 | % | ALA4028155 | % | Homo sapiens |
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