# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2181939 | 2A, (Rp isomer) | EC50 | = | 0.3 | uM | ALA2388104 | 6.52 | nM | Homo sapiens | ||
2. | ALA2181939 | 2A, (Rp isomer) | EC50 | 0 | ALA2390599 | Not Active | Homo sapiens | |||||
3. | ALA2181939 | 2A, (Rp isomer) | IC50 | = | 47 | uM | ALA2390597 | 4.33 | nM | |||
4. | ALA2181939 | 2A, (Rp isomer) | IC50 | = | 26 | uM | ALA2390596 | 4.58 | nM | |||
5. | ALA2181939 | 2A, (Rp isomer) | IC50 | = | 1 | uM | ALA2390594 | 6.00 | nM | Rattus norvegicus | ||
6. | ALA2181939 | 2A, (Rp isomer) | Drug metabolism | = | 5.4 | % | ALA2390592 | % | Homo sapiens | |||
7. | ALA2181939 | 2A, (Rp isomer) | Drug metabolism | = | 3.6 | % | ALA2390591 | % | Homo sapiens | |||
8. | ALA2181939 | 2A, (Rp isomer) | Drug metabolism | 0 | ALA2390590 | Not Determined | Homo sapiens | |||||
9. | ALA2181939 | 2A, (Rp isomer) | Drug metabolism | 0 | ALA2390589 | Not Determined | Homo sapiens | |||||
10. | ALA2181939 | 2A, (Rp isomer) | Drug metabolism | 0 | ALA2390588 | Not Determined | Homo sapiens | |||||
11. | ALA2181939 | 2A, (Rp isomer) | Drug metabolism | 0 | ALA2390587 | Not Determined | Homo sapiens | |||||
12. | ALA2181939 | 2A, (Rp isomer) | Stability | = | 56 | % | ALA2390586 | % | Homo sapiens | |||
13. | ALA2181939 | 2A, (Rp isomer) | EC50 | = | 0.22 | uM | ALA2188788 | 6.66 | nM | Meleagris gallopavo | ||
14. | ALA2181939 | 2A, (Rp isomer) | Drug metabolism | = | 5 | % | ALA2182177 | % | Homo sapiens | |||
15. | ALA2181939 | 2A, (Rp isomer) | t1/2 | = | 3.5 | hr | ALA2188784 | hr | Homo sapiens | |||
16. | ALA2181939 | 2A, (Rp isomer) | t1/2 | = | 4.2 | hr | ALA2188792 | hr |