# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2203836 | 34 | IC50 | = | 12 | nM | ALA2216251 | 7.92 | nM | Homo sapiens | ||
2. | ALA2203836 | 34 | Activity | 0 | ALA2216246 | Non-toxic | Salmonella enterica subsp. enterica serovar Typhimurium | |||||
3. | ALA2203836 | 34 | Activity | 0 | ALA2216245 | Non-toxic | Salmonella enterica subsp. enterica serovar Typhimurium | |||||
4. | ALA2203836 | 34 | Activity | 0 | ALA2216242 | Not Active | Homo sapiens | |||||
5. | ALA2203836 | 34 | IC50 | > | 10000 | nM | ALA2215818 | nM | Homo sapiens | |||
6. | ALA2203836 | 34 | Activity | 0 | ALA2214346 | Not Active | Homo sapiens | |||||
7. | ALA2203836 | 34 | Activity | 0 | ALA2214345 | Not Active | Homo sapiens | |||||
8. | ALA2203836 | 34 | Activity | = | 20 | % | ALA2214344 | % | Homo sapiens | |||
9. | ALA2203836 | 34 | IC50 | = | 11.7 | nM | ALA2214343 | 7.93 | nM | Homo sapiens | ||
10. | ALA2203836 | 34 | IC50 | = | 100 | nM | ALA2214342 | 7.00 | nM | Homo sapiens | ||
11. | ALA2203836 | 34 | Activity | 0 | ALA2214339 | Not Active | Homo sapiens | |||||
12. | ALA2203836 | 34 | Activity | = | 70 | % | ALA2214338 | % | Homo sapiens | |||
13. | ALA2203836 | 34 | Activity | = | 60 | % | ALA2214337 | % | Homo sapiens | |||
14. | ALA2203836 | 34 | Fu | = | 0.3 | % | ALA2216253 | Homo sapiens | ||||
15. | ALA2203836 | 34 | Fu | = | 1.9 | % | ALA2214336 | Rattus norvegicus | ||||
16. | ALA2203836 | 34 | CL | = | 2 | ml/min.kg | ALA2214335 | mL.min-1.kg-1 | Macaca fascicularis | |||
17. | ALA2203836 | 34 | Vdss | = | 0.3 | L/Kg | ALA2214334 | L.kg-1 | Macaca fascicularis | |||
18. | ALA2203836 | 34 | t1/2 | = | 2.8 | hr | ALA2216244 | hr | Macaca fascicularis | |||
19. | ALA2203836 | 34 | AUC | = | 18035 | ng.hr/ml | ALA2214333 | ng.hr.mL-1 | Macaca fascicularis | |||
20. | ALA2203836 | 34 | Cmax | = | 5102 | ng/ml | ALA2216252 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Macaca fascicularis |