# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2204998 | 3, GSK926 | Ki(app) | = | 7.9 | nM | ALA2209121 | 8.10 | nM | Homo sapiens | ||
2. | ALA2204998 | 3, GSK926 | IC50 | = | 0.02 | uM | ALA2209122 | 7.70 | nM | Homo sapiens | ||
3. | ALA2204998 | 3, GSK926 | IC50 | = | 2.5 | uM | ALA2209120 | 5.60 | nM | Homo sapiens | ||
4. | ALA2204998 | 3, GSK926 | IC50 | > | 100 | uM | ALA2209119 | nM | Homo sapiens | |||
5. | ALA2204998 | 3, GSK926 | IC50 | > | 100 | uM | ALA2209118 | nM | Homo sapiens | |||
6. | ALA2204998 | 3, GSK926 | IC50 | > | 100 | uM | ALA2209117 | nM | Mus musculus | |||
7. | ALA2204998 | 3, GSK926 | IC50 | > | 100 | uM | ALA2209116 | nM | Homo sapiens | |||
8. | ALA2204998 | 3, GSK926 | IC50 | > | 100 | uM | ALA2209115 | nM | Homo sapiens | |||
9. | ALA2204998 | 3, GSK926 | IC50 | > | 100 | uM | ALA2209110 | nM | Homo sapiens | |||
10. | ALA2204998 | 3, GSK926 | IC50 | > | 100 | uM | ALA2209109 | nM | Homo sapiens | |||
11. | ALA2204998 | 3, GSK926 | IC50 | > | 100 | uM | ALA2209108 | nM | Homo sapiens | |||
12. | ALA2204998 | 3, GSK926 | IC50 | > | 100 | uM | ALA2209107 | nM | Homo sapiens | |||
13. | ALA2204998 | 3, GSK926 | IC50 | = | 214 | uM | ALA2209106 | nM | Homo sapiens | |||
14. | ALA2204998 | 3, GSK926 | IC50 | > | 100 | uM | ALA2209105 | nM | Homo sapiens | |||
15. | ALA2204998 | 3, GSK926 | IC50 | > | 100 | uM | ALA2209104 | nM | Homo sapiens | |||
16. | ALA2204998 | 3, GSK926 | IC50 | > | 100 | uM | ALA2209077 | nM | Homo sapiens | |||
17. | ALA2204998 | 3, GSK926 | IC50 | = | 324 | nM | ALA2209076 | 6.49 | nM | Homo sapiens | ||
18. | ALA2204998 | 3, GSK926 | INH | 0 | ALA2209076 | Dose-dependent effect | % | Homo sapiens | ||||
19. | ALA2204998 | 3, GSK926 | INH | > | 90 | % | ALA2209075 | % | Homo sapiens | |||
20. | ALA2204998 | 3, GSK926 | INH | 0 | ALA2209074 | Active | % | Homo sapiens |