| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA2207081 | 14 | pIC50 | < | 4.3 | ALA2212599 | nM | Homo sapiens | ||||
| 2. | ALA2207081 | 14 | pIC50 | < | 4.3 | ALA2212601 | nM | Homo sapiens | ||||
| 3. | ALA2207081 | 14 | Activity | = | -7 | % | ALA2214986 | % | Mus musculus | |||
| 4. | ALA2207081 | 14 | t1/2 | = | 0.7 | hr | ALA2212603 | hr | Rattus norvegicus | |||
| 5. | ALA2207081 | 14 | t1/2 | = | 0.7 | hr | ALA2212586 | hr | Mus musculus | |||
| 6. | ALA2207081 | 14 | logD | = | 2.6 | ALA2212606 | ||||||
| 7. | ALA2207081 | 14 | AUC | = | 2.9 | hr.microg/ml | ALA2212591 | ng.hr.mL-1 | Mus musculus | |||
| 8. | ALA2207081 | 14 | AUC | = | 3.7 | hr.microg/ml | ALA2212592 | ng.hr.mL-1 | Mus musculus | |||
| 9. | ALA2207081 | 14 | CL | = | 4.5 | ml/min.kg | ALA2212587 | mL.min-1.kg-1 | Mus musculus | |||
| 10. | ALA2207081 | 14 | pA2 | = | 5 | ALA2212593 | 5.00 | nM | Homo sapiens | |||
| 11. | ALA2207081 | 14 | pIC50 | = | 5.4 | ALA2214982 | 5.40 | nM | Homo sapiens | |||
| 12. | ALA2207081 | 14 | pKi | < | 5.7 | ALA2212596 | nM | Mus musculus | ||||
| 13. | ALA2207081 | 14 | pKa | = | 5.9 | ALA2212605 | ||||||
| 14. | ALA2207081 | 14 | pIC50 | = | 6.2 | ALA2212598 | 6.20 | nM | Homo sapiens | |||
| 15. | ALA2207081 | 14 | pKi | = | 6.4 | ALA2213078 | 6.40 | nM | Homo sapiens | |||
| 16. | ALA2207081 | 14 | pKi | = | 6.4 | ALA2213077 | 6.40 | nM | Homo sapiens | |||
| 17. | ALA2207081 | 14 | pIC50 | = | 6.7 | ALA2212600 | 6.70 | nM | Homo sapiens | |||
| 18. | ALA2207081 | 14 | pKi | = | 7 | ALA2213075 | 7.00 | nM | Homo sapiens | |||
| 19. | ALA2207081 | 14 | pKi | = | 7.1 | ALA2213076 | 7.10 | nM | Homo sapiens | |||
| 20. | ALA2207081 | 14 | pKi | = | 8 | ALA2213079 | 8.00 | nM | Homo sapiens |
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