| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA2207429 | 10e | beta t1/2 | = | 2.2 | hr | ALA2209555 | hr | Rattus norvegicus | |||
| 2. | ALA2207429 | 10e | CL | = | 3.2 | ml/min.kg | ALA2209542 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 3. | ALA2207429 | 10e | CLH | = | 53 | ml/min.kg | ALA2209548 | mL.min-1.kg-1 | Homo sapiens | |||
| 4. | ALA2207429 | 10e | Cmax | = | 38265 | nM | ALA2209540 | nM | Rattus norvegicus | |||
| 5. | ALA2207429 | 10e | F | = | 69 | % | ALA2209538 | % | Rattus norvegicus | |||
| 6. | ALA2207429 | 10e | fCmax | = | 25 | nM | ALA2209539 | nM | Rattus norvegicus | |||
| 7. | ALA2207429 | 10e | Fu | = | 0.001 | ALA2209537 | Rattus norvegicus | |||||
| 8. | ALA2207429 | 10e | IC50 | > | 10000 | nM | ALA2209546 | nM | Homo sapiens | |||
| 9. | ALA2207429 | 10e | IC50 | = | 398 | nM | ALA2209550 | 6.40 | nM | Homo sapiens | ||
| 10. | ALA2207429 | 10e | IC50 | = | 553 | nM | ALA2209549 | 6.26 | nM | Mus musculus | ||
| 11. | ALA2207429 | 10e | INH | = | 31 | % | ALA2209547 | % | Homo sapiens | |||
| 12. | ALA2207429 | 10e | INH | 0 | ALA2209543 | Not Active | % | Homo sapiens | ||||
| 13. | ALA2207429 | 10e | Vdss | = | 0.4 | L/Kg | ALA2209541 | L.kg-1 | Rattus norvegicus |
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