| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA2207441 | 13k | beta t1/2 | = | 7.3 | hr | ALA2209536 | hr | Rattus norvegicus | |||
| 2. | ALA2207441 | 13k | CLH | = | 149 | ml/min.kg | ALA2209548 | mL.min-1.kg-1 | Homo sapiens | |||
| 3. | ALA2207441 | 13k | Cmax | = | 68 | nM | ALA2209535 | nM | Rattus norvegicus | |||
| 4. | ALA2207441 | 13k | fCmax | = | 1.1 | nM | ALA2209534 | nM | Rattus norvegicus | |||
| 5. | ALA2207441 | 13k | Fu | = | 0.016 | ALA2209537 | Rattus norvegicus | |||||
| 6. | ALA2207441 | 13k | IC50 | = | 12.5 | nM | ALA2209550 | 7.90 | nM | Homo sapiens | ||
| 7. | ALA2207441 | 13k | IC50 | = | 62 | nM | ALA2209549 | 7.21 | nM | Mus musculus | ||
| 8. | ALA2207441 | 13k | IC50 | = | 473 | nM | ALA2209546 | 6.33 | nM | Homo sapiens | ||
| 9. | ALA2207441 | 13k | INH | = | 12 | % | ALA2209547 | % | Homo sapiens | |||
| 10. | ALA2207441 | 13k | INH | 0 | ALA2209543 | Not Active | % | Homo sapiens | ||||
| 11. | ALA2207441 | 13k | logD | = | 4.7 | ALA2209551 |
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