| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA2216902 | 15 | LogD7.4 | 2.9 | ALA3301363 | |||||||
| 2. | ALA2216902 | 15 | CLint | 20.42 | microL/min/mg | ALA3301370 | mL.min-1.g-1 | |||||
| 3. | ALA2216902 | 15 | PPB | 78.01 | % | ALA3301366 | % | |||||
| 4. | ALA2216902 | 15 | PPB | 78.01 | % | ALA3301365 | % | |||||
| 5. | ALA2216902 | 15 | CLint | 10 | microL/min/1E6 cells | ALA3301371 | uL.min-1.(10^6cells)-1 | |||||
| 6. | ALA2216902 | 15 | Ki | = | 0 | uM | ALA2217262 | 9.34 | nM | Homo sapiens | ||
| 7. | ALA2216902 | 15 | Ratio Ki | = | 256 | ALA2217279 | ||||||
| 8. | ALA2216902 | 15 | IC50 | = | 0.003 | uM | ALA2217317 | 8.52 | nM | Homo sapiens | ||
| 9. | ALA2216902 | 15 | Ki(app) | = | 0.47 | nM | ALA2415771 | 9.33 | nM | Homo sapiens | ||
| 10. | ALA2216902 | 15 | Ratio Ki(app) | = | 256 | ALA2415769 | ||||||
| 11. | ALA2216902 | 15 | IC50 | = | 4.38 | nM | ALA2415716 | 8.36 | nM | Homo sapiens | ||
| 12. | ALA2216902 | 15 | Ratio Ki(app) | = | 420 | ALA2415715 | ||||||
| 13. | ALA2216902 | 15 | Ratio Ki(app) | = | 219 | ALA2415714 | ||||||
| 14. | ALA2216902 | 15 | INH | = | 61 | % | ALA2415713 | % | Homo sapiens | |||
| 15. | ALA2216902 | 15 | INH | = | 71 | % | ALA2415712 | % | Homo sapiens | |||
| 16. | ALA2216902 | 15 | CLH | = | 1.4 | ml/min.kg | ALA2415710 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 17. | ALA2216902 | 15 | CLH | = | 6.2 | ml/min.kg | ALA2415711 | mL.min-1.kg-1 | ||||
| 18. | ALA2216902 | 15 | PPB | = | 81.7 | % | ALA2415709 | % | Rattus norvegicus | |||
| 19. | ALA2216902 | 15 | PPB | = | 80 | % | ALA2415708 | % | Canis lupus familiaris | |||
| 20. | ALA2216902 | 15 | CL | = | 19.4 | ml/min.kg | ALA2415706 | mL.min-1.kg-1 | Rattus norvegicus |
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