# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | AG-1024 | Tyrphostin AG-1024 | IC50 relative | = | 7.206 | uM | ALA5303712 | Active | uM | Severe acute respiratory syndrome coronavirus 2 | ||
2. | AG-1024 | Tyrphostin AG-1024 | INH | = | 80 | % | ALA3365632 | % | Homo sapiens | |||
3. | AG-1024 | Tyrphostin AG-1024 | Selectivity index | = | 1.18 | ALA4513085 | Selectivity Index = Cc50/Ic50 | |||||
4. | AG-1024 | Tyrphostin AG-1024 | CC50 | = | 10.37 | uM | ALA4513084 | nM | Chlorocebus sabaeus | |||
5. | AG-1024 | Tyrphostin AG-1024 | IC50 | = | 8.77 | uM | ALA4513083 | 5.06 | nM | Severe acute respiratory syndrome coronavirus 2 | ||
6. | AG-1024 | Tyrphostin AG-1024 | inhibition | = | 36.93 | % | ALA4513082 | % | Severe acute respiratory syndrome coronavirus 2 | |||
7. | AG-1024 | Tyrphostin AG-1024 | inhibition | = | 47.67 | % | ALA4513082 | % | Severe acute respiratory syndrome coronavirus 2 | |||
8. | AG-1024 | Tyrphostin AG-1024 | Inhibition | = | 6.898 | % | ALA4495582 | % | Severe acute respiratory syndrome coronavirus 2 | |||
9. | AG-1024 | Tyrphostin AG-1024 | Inhibition | = | 11.19 | % | ALA4495582 | % | Severe acute respiratory syndrome coronavirus 2 | |||
10. | AG-1024 | Tyrphostin AG-1024 | CC50 | = | 10.37 | uM | ALA4513084 | nM | Chlorocebus sabaeus | |||
11. | AG-1024 | Tyrphostin AG-1024 | IC50 | = | 8.77 | uM | ALA4513083 | 5.06 | nM | Severe acute respiratory syndrome coronavirus 2 | ||
12. | AG-1024 | Tyrphostin AG-1024 | Selectivity index | = | 1.18 | ALA4513085 | Selectivity Index = Cc50/Ic50 | |||||
13. | AG-1024 | Tyrphostin AG-1024 | inhibition | = | 36.93 | % | ALA4513082 | % | Severe acute respiratory syndrome coronavirus 2 | |||
14. | AG-1024 | Tyrphostin AG-1024 | inhibition | = | 47.67 | % | ALA4513082 | % | Severe acute respiratory syndrome coronavirus 2 | |||
15. | AG-1024 | Tyrphostin AG-1024 | inhibition | = | 2.56 | % | ALA4808150 | % | Homo sapiens | |||
16. | AG-1024 | Tyrphostin AG-1024 | inhibition | = | 8.73 | % | ALA4808149 | % | Homo sapiens | |||
17. | AG-1024 | Tyrphostin AG-1024 | Inhibition | = | -2.54 | % | ALA4303805 | % | Severe acute respiratory syndrome coronavirus 2 | |||
18. | AG-1024 | Tyrphostin AG-1024 | KD | = | 0 | M | ALA3885749 | 7.15 | nM | Homo sapiens | ||
19. | AG-1024 | Tyrphostin AG-1024 | kon | = | 407000 | Ms-1 | ALA3885749 | Ms-1 | Homo sapiens | |||
20. | AG-1024 | Tyrphostin AG-1024 | koff | = | 0.029 | s-1 | ALA3885749 | s-1 | Homo sapiens |