| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  A 61603 hydrobromide | A-61603 | pKi | = | 7.92 | ALA3056712 | 7.92 | nM | Rattus norvegicus | |||
| 2. | A 61603 hydrobromide | A-61603 | pKi | = | 5.53 | ALA3056713 | 5.53 | nM | Mesocricetus auratus | |||
| 3. | A 61603 hydrobromide | A-61603 | pKi | = | 5.83 | ALA3056710 | 5.83 | nM | Rattus norvegicus | |||
| 4. | A 61603 hydrobromide | A-61603 | pEC50 | = | 8.03 | ALA3056711 | 8.03 | nM | Oryctolagus cuniculus | |||
| 5. | A 61603 hydrobromide | A-61603 | Efficacy | = | 88 | % | ALA3057222 | % | Oryctolagus cuniculus | |||
| 6. | A 61603 hydrobromide | A-61603 | pEC50 | = | 6.5 | ALA3056709 | 6.50 | nM | Rattus norvegicus | |||
| 7. | A 61603 hydrobromide | A-61603 | Efficacy | = | 91 | % | ALA3057220 | % | Rattus norvegicus | |||
| 8. | A 61603 hydrobromide | A-61603 | pEC50 | = | 5.59 | ALA3057221 | 5.59 | nM | Rattus norvegicus | |||
| 9. | A 61603 hydrobromide | A-61603 | Efficacy | = | 99 | % | ALA3057219 | % | Rattus norvegicus | |||
| 10. | A 61603 hydrobromide | A-61603 | Selectivity Index | = | 1.7 | ALA3057217 | Canis lupus familiaris | |||||
| 11. | A 61603 hydrobromide | A-61603 | pKi | = | 7.48 | ALA3057218 | 7.48 | nM | Homo sapiens | |||
| 12. | A 61603 hydrobromide | A-61603 | pKi | = | 6.61 | ALA3057215 | 6.61 | nM | Rattus norvegicus | |||
| 13. | A 61603 hydrobromide | A-61603 | Delta TM | = | -2.47 | C | ALA5068376 | Thermal Shift Assay | C | Homo sapiens | ||
| 14. | A 61603 hydrobromide | A-61603 | Delta TM | = | 0.42 | C | ALA5066518 | Thermal Shift Assay | C | Homo sapiens | ||
| 15. | A 61603 hydrobromide | A-61603 | Delta TM | = | -0.14 | C | ALA5065589 | Thermal Shift Assay | C | Homo sapiens | ||
| 16. | A 61603 hydrobromide | A-61603 | Delta TM | = | 0.4 | C | ALA5064660 | Thermal Shift Assay | C | Homo sapiens | ||
| 17. | A 61603 hydrobromide | A-61603 | Delta TM | = | 0.49 | C | ALA5063731 | Thermal Shift Assay | C | Homo sapiens | ||
| 18. | A 61603 hydrobromide | A-61603 | Delta TM | = | 0.32 | C | ALA5062802 | Thermal Shift Assay | C | Homo sapiens | ||
| 19. | A 61603 hydrobromide | A-61603 | Delta TM | = | -4.67 | C | ALA4650107 | Thermal Shift Assay | C | Homo sapiens | ||
| 20. | A 61603 hydrobromide | A-61603 | Delta TM | = | -3.21 | C | ALA5060944 | Thermal Shift Assay | C | Homo sapiens |
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