# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA94219 | Gemini | Ratio IC50 | = | 0.1 | ALA917204 | ||||||
2. | ALA94219 | Gemini | Stability | = | 80 | % | ALA917195 | % | Rattus norvegicus | |||
3. | ALA94219 | Gemini | IC50 | = | 4 | pM | ALA917203 | nM | ||||
4. | ALA94219 | Gemini | MTD | < | 1 | mg kg-1 | ALA917202 | mg kg-1 | Mus musculus | |||
5. | ALA94219 | Gemini | Drug uptake | = | 16.73 | mg kg-1 | ALA917199 | mg kg-1 | Mus musculus | |||
6. | ALA94219 | Gemini | Drug uptake | = | 12.3 | mg kg-1 | ALA917198 | mg kg-1 | Mus musculus | |||
7. | ALA94219 | Gemini | Drug uptake | = | 11.07 | mg kg-1 | ALA917197 | mg kg-1 | Mus musculus | |||
8. | ALA94219 | Gemini | ED50 | = | 82 | nM | ALA709609 | 7.09 | nM | Homo sapiens | ||
9. | ALA94219 | Gemini | ED50 | = | 1.2 | nM | ALA707645 | 8.92 | nM | Homo sapiens | ||
10. | ALA94219 | Gemini | ED50 | = | 0.34 | nM | ALA693704 | 9.47 | nM | Homo sapiens | ||
11. | ALA94219 | Gemini | ED50 | = | 180 | nM | ALA848190 | 6.75 | nM | |||
12. | ALA94219 | Gemini | ED50 | = | 1 | nM | ALA770791 | 9.00 | nM | |||
13. | ALA94219 | Gemini | RCI | = | 38 | % | ALA820134 | % | Gallus gallus | |||
14. | ALA94219 | Gemini | RCI | = | 2.5 | % | ALA818848 | % | Homo sapiens |