# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | MeOSuc-AAPV-CMK | 39 N-(methoxysuccinyl)-L-Ala-L-Ala-L-Pro-L-Val Chloromethyl ketone | Activity | = | 50 | % | ALA4713853 | % | Mus musculus | |||
2. | MeOSuc-AAPV-CMK | 39 N-(methoxysuccinyl)-L-Ala-L-Ala-L-Pro-L-Val Chloromethyl ketone | Activity | 0 | ALA4713852 | Active | Mus musculus | |||||
3. | MeOSuc-AAPV-CMK | 39 N-(methoxysuccinyl)-L-Ala-L-Ala-L-Pro-L-Val Chloromethyl ketone | Activity | 0 | ALA4713851 | Non-Toxic | ||||||
4. | MeOSuc-AAPV-CMK | 39 N-(methoxysuccinyl)-L-Ala-L-Ala-L-Pro-L-Val Chloromethyl ketone | Activity | 0 | ALA4713849 | Dose-dependent effect | ||||||
5. | MeOSuc-AAPV-CMK | 39 N-(methoxysuccinyl)-L-Ala-L-Ala-L-Pro-L-Val Chloromethyl ketone | INH | 0 | ALA4713847 | Dose-dependent effect | % | |||||
6. | MeOSuc-AAPV-CMK | 39 N-(methoxysuccinyl)-L-Ala-L-Ala-L-Pro-L-Val Chloromethyl ketone | IC50 | = | 2.74 | uM | ALA4713847 | 5.56 | nM | |||
7. | MeOSuc-AAPV-CMK | 39 N-(methoxysuccinyl)-L-Ala-L-Ala-L-Pro-L-Val Chloromethyl ketone | INH | = | 23.2 | % | ALA5041633 | % | ||||
8. | MeOSuc-AAPV-CMK | 39 N-(methoxysuccinyl)-L-Ala-L-Ala-L-Pro-L-Val Chloromethyl ketone | IC50 | = | 0.5 | mM | ALA762661 | nM | Sus scrofa |