# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | WAY-659977 | 4 | IC50 | = | 0.008 | uM | ALA2317531 | 8.10 | nM | Homo sapiens | ||
2. | WAY-659977 | 4 | IC50 | = | 0.002 | uM | ALA2317530 | 8.70 | nM | Homo sapiens | ||
3. | WAY-659977 | 4 | IC50 | = | 0.931 | uM | ALA2317529 | 6.03 | nM | Homo sapiens | ||
4. | WAY-659977 | 4 | Ratio IC50 | > | 100 | ALA2317527 | ||||||
5. | WAY-659977 | 4 | IC50 | = | 36 | uM | ALA2317528 | 4.44 | nM | Homo sapiens | ||
6. | WAY-659977 | 4 | t1/2 | = | 40 | min | ALA5227348 | hr | ||||
7. | WAY-659977 | 4 | IC50 | = | 160 | nM | ALA5227346 | 6.80 | nM | |||
8. | WAY-659977 | 4 | IC50 | = | 2 | nM | ALA5227343 | 8.70 | nM | Homo sapiens | ||
9. | WAY-659977 | 4 | IC50 | = | 8 | nM | ALA5227342 | 8.10 | nM | Homo sapiens | ||
10. | WAY-659977 | 4 | IC50 | = | 0.01 | uM | ALA3111843 | 8.00 | nM | Homo sapiens | ||
11. | WAY-659977 | 4 | IC50 | = | 0.16 | uM | ALA3111842 | 6.80 | nM | |||
12. | WAY-659977 | 4 | t1/2 | = | 35 | min | ALA3111840 | hr | Mus musculus | |||
13. | WAY-659977 | 4 | solubility | = | 6.6 | ug ml-1 | ALA3111839 | ug.mL-1 | ||||
14. | WAY-659977 | 4 | Vdss | = | 4.69 | L/Kg | ALA3111846 | L.kg-1 | Rattus norvegicus | |||
15. | WAY-659977 | 4 | t1/2 | = | 0.37 | hr | ALA3111847 | hr | Rattus norvegicus | |||
16. | WAY-659977 | 4 | AUC | = | 0.11 | uM.hr | ALA3111849 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
17. | WAY-659977 | 4 | CL | = | 10.9 | L/hr/kg | ALA3111848 | mL.min-1.kg-1 | Rattus norvegicus |