# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2324411 | SI-4, R248C1 | Ratio IC50 | = | 4 | ALA4040179 | ||||||
2. | ALA2324411 | SI-4, R248C1 | Ratio IC50 | = | 9 | ALA4040178 | ||||||
3. | ALA2324411 | SI-4, R248C1 | Ratio IC50 | = | 7 | ALA4040177 | ||||||
4. | ALA2324411 | SI-4, R248C1 | pKa | = | 3.5 | ALA4040145 | ||||||
5. | ALA2324411 | SI-4, R248C1 | CLH(app) | > | 262 | microL/min/mg | ALA4040134 | mL.min-1.g-1 | Homo sapiens | |||
6. | ALA2324411 | SI-4, R248C1 | IC50 | 0 | ALA4040133 | Not Determined | Homo sapiens | |||||
7. | ALA2324411 | SI-4, R248C1 | IC50 | 0 | ALA4040132 | Not Determined | Homo sapiens | |||||
8. | ALA2324411 | SI-4, R248C1 | IC50 | = | 124 | nM | ALA4040131 | 6.91 | nM | Rattus norvegicus | ||
9. | ALA2324411 | SI-4, R248C1 | IC50 | > | 3000 | nM | ALA4040130 | nM | Homo sapiens | |||
10. | ALA2324411 | SI-4, R248C1 | IC50 | = | 510 | nM | ALA4040129 | 6.29 | nM | Homo sapiens | ||
11. | ALA2324411 | SI-4, R248C1 | IC50 | = | 292 | nM | ALA4040128 | 6.54 | nM | Homo sapiens | ||
12. | ALA2324411 | SI-4, R248C1 | IC50 | = | 149 | nM | ALA4040127 | 6.83 | nM | Homo sapiens | ||
13. | ALA2324411 | SI-4, R248C1 | IC50 | = | 216 | nM | ALA4040126 | 6.67 | nM | Homo sapiens | ||
14. | ALA2324411 | SI-4, R248C1 | IC50 | = | 31 | nM | ALA4040125 | 7.51 | nM | Homo sapiens | ||
15. | ALA2324411 | SI-4, R248C1 | IC50 | = | 15060 | nM | ALA4040124 | 4.82 | nM | Homo sapiens | ||
16. | ALA2324411 | SI-4, R248C1 | pIC50 | = | 7.444 | ALA2328568 | 7.44 | nM | Homo sapiens |