# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2324753 | SI-4, R180C1 | Ratio IC50 | = | 39 | ALA4040179 | ||||||
2. | ALA2324753 | SI-4, R180C1 | Ratio IC50 | > | 140 | ALA4040178 | ||||||
3. | ALA2324753 | SI-4, R180C1 | Ratio IC50 | > | 140 | ALA4040177 | ||||||
4. | ALA2324753 | SI-4, R180C1 | pKa | = | 3.5 | ALA4040145 | ||||||
5. | ALA2324753 | SI-4, R180C1 | CLH(app) | = | 92 | microL/min/mg | ALA4040134 | mL.min-1.g-1 | Homo sapiens | |||
6. | ALA2324753 | SI-4, R180C1 | IC50 | = | 517 | nM | ALA4040133 | 6.29 | nM | Homo sapiens | ||
7. | ALA2324753 | SI-4, R180C1 | IC50 | = | 556 | nM | ALA4040132 | 6.25 | nM | Homo sapiens | ||
8. | ALA2324753 | SI-4, R180C1 | IC50 | = | 813 | nM | ALA4040131 | 6.09 | nM | Rattus norvegicus | ||
9. | ALA2324753 | SI-4, R180C1 | IC50 | > | 10000 | nM | ALA4040130 | nM | Homo sapiens | |||
10. | ALA2324753 | SI-4, R180C1 | IC50 | = | 199 | nM | ALA4040129 | 6.70 | nM | Homo sapiens | ||
11. | ALA2324753 | SI-4, R180C1 | IC50 | > | 3000 | nM | ALA4040128 | nM | Homo sapiens | |||
12. | ALA2324753 | SI-4, R180C1 | IC50 | = | 276 | nM | ALA4040127 | 6.56 | nM | Homo sapiens | ||
13. | ALA2324753 | SI-4, R180C1 | IC50 | > | 3000 | nM | ALA4040126 | nM | Homo sapiens | |||
14. | ALA2324753 | SI-4, R180C1 | IC50 | = | 21 | nM | ALA4040125 | 7.68 | nM | Homo sapiens | ||
15. | ALA2324753 | SI-4, R180C1 | IC50 | > | 30000 | nM | ALA4040124 | nM | Homo sapiens | |||
16. | ALA2324753 | SI-4, R180C1 | pIC50 | = | 7.699 | ALA2328568 | 7.70 | nM | Homo sapiens |