| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA2325485 | 9b, ML299 | IC50 | = | 6 | nM | ALA2330403 | 8.22 | nM | Homo sapiens | ||
| 2. | ALA2325485 | 9b, ML299 | IC50 | = | 20 | nM | ALA2330327 | 7.70 | nM | Homo sapiens | ||
| 3. | ALA2325485 | 9b, ML299 | IC50 | = | 48 | nM | ALA2330326 | 7.32 | nM | Homo sapiens | ||
| 4. | ALA2325485 | 9b, ML299 | IC50 | = | 84 | nM | ALA2330325 | 7.08 | nM | Homo sapiens | ||
| 5. | ALA2325485 | 9b, ML299 | Stability | 0 | ALA2330324 | Stable | % | |||||
| 6. | ALA2325485 | 9b, ML299 | solubility | 0 | ALA2330322 | soluble | ||||||
| 7. | ALA2325485 | 9b, ML299 | INH | > | 50 | % | ALA2330323 | % | Homo sapiens | |||
| 8. | ALA2325485 | 9b, ML299 | INH | > | 50 | % | ALA2330321 | % | Homo sapiens | |||
| 9. | ALA2325485 | 9b, ML299 | INH | > | 50 | % | ALA2330320 | % | Homo sapiens | |||
| 10. | ALA2325485 | 9b, ML299 | IC50 | > | 20 | uM | ALA2330319 | nM | Homo sapiens | |||
| 11. | ALA2325485 | 9b, ML299 | CLH | = | 61.8 | ml/min.kg | ALA2330317 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 12. | ALA2325485 | 9b, ML299 | CLH | = | 19.1 | ml/min.kg | ALA2330318 | mL.min-1.kg-1 | Homo sapiens | |||
| 13. | ALA2325485 | 9b, ML299 | IC50 | > | 30 | uM | ALA2330316 | nM | Homo sapiens | |||
| 14. | ALA2325485 | 9b, ML299 | IC50 | = | 13.3 | uM | ALA2330313 | 4.88 | nM | Homo sapiens | ||
| 15. | ALA2325485 | 9b, ML299 | IC50 | = | 6.8 | uM | ALA2330314 | 5.17 | nM | Homo sapiens | ||
| 16. | ALA2325485 | 9b, ML299 | IC50 | = | 9.4 | uM | ALA2330315 | 5.03 | nM | Homo sapiens | ||
| 17. | ALA2325485 | 9b, ML299 | Fu | = | 3 | % | ALA2330311 | Rattus norvegicus | ||||
| 18. | ALA2325485 | 9b, ML299 | Fu | = | 1 | % | ALA2330312 | Homo sapiens | ||||
| 19. | ALA2325485 | 9b, ML299 | Cp | = | 1.08 | uM.hr | ALA2330308 | uM.hr | Mus musculus | |||
| 20. | ALA2325485 | 9b, ML299 | AUC | = | 48.5 | uM.hr | ALA2330309 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Mus musculus |
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