# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2332056 | 14b | t1/2 | > | 120 | min | ALA2341181 | hr | Homo sapiens | |||
2. | ALA2332056 | 14b | IC50 | > | 20 | uM | ALA2341178 | nM | Homo sapiens | |||
3. | ALA2332056 | 14b | IC50 | > | 20 | uM | ALA2341177 | nM | Homo sapiens | |||
4. | ALA2332056 | 14b | INH | = | -2 | % | ALA2341175 | % | Homo sapiens | |||
5. | ALA2332056 | 14b | Vd | = | 0.7 | L/Kg | ALA2341166 | L.kg-1 | Rattus norvegicus | |||
6. | ALA2332056 | 14b | IC50 | = | 2 | nM | ALA2341182 | 8.70 | nM | Homo sapiens | ||
7. | ALA2332056 | 14b | t1/2 | = | 2.1 | hr | ALA2341165 | hr | Rattus norvegicus | |||
8. | ALA2332056 | 14b | CL | = | 4.9 | ml/min.kg | ALA2341167 | mL.min-1.kg-1 | Rattus norvegicus | |||
9. | ALA2332056 | 14b | Cmax | = | 9.2 | uM | ALA2341163 | nM | Rattus norvegicus | |||
10. | ALA2332056 | 14b | AUC | = | 9.5 | uM.hr | ALA2341164 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
11. | ALA2332056 | 14b | IC50 | = | 10 | nM | ALA2341176 | 8.00 | nM | Homo sapiens | ||
12. | ALA2332056 | 14b | INH | = | 23 | % | ALA2341172 | % | Homo sapiens | |||
13. | ALA2332056 | 14b | F | = | 28 | % | ALA2341162 | % | Rattus norvegicus | |||
14. | ALA2332056 | 14b | IC50 | = | 32 | nM | ALA2341183 | 7.50 | nM | |||
15. | ALA2332056 | 14b | INH | = | 41 | % | ALA2341173 | % | Homo sapiens | |||
16. | ALA2332056 | 14b | INH | = | 71 | % | ALA2341174 | % | Homo sapiens | |||
17. | ALA2332056 | 14b | IC50 | = | 580 | nM | ALA2341180 | 6.24 | nM | |||
18. | ALA2332056 | 14b | IC50 | = | 6400 | nM | ALA2341179 | 5.19 | nM | Homo sapiens | ||
19. | ALA2332056 | 14b | pIC50 | = | 8.699 | ALA3404496 | 8.70 | nM | Homo sapiens | |||
20. | ALA2332056 | 14b | IC50 | = | 580 | nM | ALA3404497 | 6.24 | nM |