| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA2332065 | 12e | IC50 | > | 100 | uM | ALA2341171 | nM | Homo sapiens | |||
| 2. | ALA2332065 | 12e | IC50 | > | 20 | uM | ALA2341178 | nM | Homo sapiens | |||
| 3. | ALA2332065 | 12e | IC50 | > | 20 | uM | ALA2341177 | nM | Homo sapiens | |||
| 4. | ALA2332065 | 12e | INH | = | -23 | % | ALA2341175 | % | Homo sapiens | |||
| 5. | ALA2332065 | 12e | IC50 | = | 1 | nM | ALA2341182 | 9.00 | nM | Homo sapiens | ||
| 6. | ALA2332065 | 12e | Vd | = | 1 | L/Kg | ALA2341166 | L.kg-1 | Rattus norvegicus | |||
| 7. | ALA2332065 | 12e | t1/2 | = | 1.6 | hr | ALA2341165 | hr | Rattus norvegicus | |||
| 8. | ALA2332065 | 12e | IC50 | = | 2 | uM | ALA2341170 | 5.70 | nM | Homo sapiens | ||
| 9. | ALA2332065 | 12e | Cmax | = | 3.8 | uM | ALA2341163 | nM | Rattus norvegicus | |||
| 10. | ALA2332065 | 12e | AUC | = | 4.2 | uM.hr | ALA2341164 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
| 11. | ALA2332065 | 12e | IC50 | = | 6 | nM | ALA2341176 | 8.22 | nM | Homo sapiens | ||
| 12. | ALA2332065 | 12e | CL | = | 11.2 | ml/min.kg | ALA2341167 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 13. | ALA2332065 | 12e | IC50 | = | 19 | nM | ALA2341183 | 7.72 | nM | |||
| 14. | ALA2332065 | 12e | t1/2 | = | 24 | min | ALA2341181 | hr | Homo sapiens | |||
| 15. | ALA2332065 | 12e | IC50 | = | 35 | uM | ALA2341168 | 4.46 | nM | Homo sapiens | ||
| 16. | ALA2332065 | 12e | INH | = | 38 | % | ALA2341173 | % | Homo sapiens | |||
| 17. | ALA2332065 | 12e | IC50 | = | 40 | uM | ALA2341169 | 4.40 | nM | Homo sapiens | ||
| 18. | ALA2332065 | 12e | F | = | 51 | % | ALA2341162 | % | Rattus norvegicus | |||
| 19. | ALA2332065 | 12e | INH | = | 95 | % | ALA2341174 | % | Homo sapiens | |||
| 20. | ALA2332065 | 12e | IC50 | = | 2988 | nM | ALA2341180 | 5.53 | nM |
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