| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA2332097 | 12a | IC50 | > | 100 | uM | ALA2341171 | nM | Homo sapiens | |||
| 2. | ALA2332097 | 12a | IC50 | > | 100 | uM | ALA2341169 | nM | Homo sapiens | |||
| 3. | ALA2332097 | 12a | IC50 | > | 100 | uM | ALA2341168 | nM | Homo sapiens | |||
| 4. | ALA2332097 | 12a | Ratio IC50 | > | 1000 | ALA2341160 | ||||||
| 5. | ALA2332097 | 12a | IC50 | > | 20 | uM | ALA2341178 | nM | Homo sapiens | |||
| 6. | ALA2332097 | 12a | IC50 | > | 20 | uM | ALA2341177 | nM | Homo sapiens | |||
| 7. | ALA2332097 | 12a | IC50 | = | 0.6 | uM | ALA2341170 | 6.22 | nM | Homo sapiens | ||
| 8. | ALA2332097 | 12a | IC50 | = | 1 | nM | ALA2341182 | 9.00 | nM | Homo sapiens | ||
| 9. | ALA2332097 | 12a | t1/2 | = | 1 | hr | ALA2341165 | hr | Rattus norvegicus | |||
| 10. | ALA2332097 | 12a | Vd | = | 1.1 | L/Kg | ALA2341166 | L.kg-1 | Rattus norvegicus | |||
| 11. | ALA2332097 | 12a | Cmax | = | 2.6 | uM | ALA2341163 | nM | Rattus norvegicus | |||
| 12. | ALA2332097 | 12a | IC50 | = | 4 | nM | ALA2341183 | 8.40 | nM | |||
| 13. | ALA2332097 | 12a | IC50 | = | 4 | nM | ALA2341176 | 8.40 | nM | Homo sapiens | ||
| 14. | ALA2332097 | 12a | AUC | = | 5.9 | uM.hr | ALA2341164 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
| 15. | ALA2332097 | 12a | INH | = | 9 | % | ALA2341175 | % | Homo sapiens | |||
| 16. | ALA2332097 | 12a | CL | = | 9.4 | ml/min.kg | ALA2341167 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 17. | ALA2332097 | 12a | t1/2 | = | 23 | min | ALA2341181 | hr | Homo sapiens | |||
| 18. | ALA2332097 | 12a | INH | = | 45 | % | ALA2341173 | % | Homo sapiens | |||
| 19. | ALA2332097 | 12a | F | = | 48 | % | ALA2341162 | % | Rattus norvegicus | |||
| 20. | ALA2332097 | 12a | INH | = | 96 | % | ALA2341174 | % | Homo sapiens |
The page will load shortly, Thanks for your patience!