# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2335071 | 1, [18F]4F-MHPG | Drug uptake | = | 0.68 | ml/min | ALA2344436 | ml/min | Rattus norvegicus | |||
2. | ALA2335071 | 1, [18F]4F-MHPG | t1/2 | > | 13 | hr | ALA2344435 | hr | Rattus norvegicus | |||
3. | ALA2335071 | 1, [18F]4F-MHPG | Drug uptake | = | 1.45 | % ID/g | ALA2344434 | % ID/g | Rattus norvegicus | |||
4. | ALA2335071 | 1, [18F]4F-MHPG | Drug uptake | = | 0.43 | % ID/g | ALA2344432 | % ID/g | Rattus norvegicus | |||
5. | ALA2335071 | 1, [18F]4F-MHPG | Drug uptake | = | 1.14 | % ID/g | ALA2344433 | % ID/g | Rattus norvegicus | |||
6. | ALA2335071 | 1, [18F]4F-MHPG | Drug uptake | = | 0.56 | % ID/g | ALA2344431 | % ID/g | Rattus norvegicus | |||
7. | ALA2335071 | 1, [18F]4F-MHPG | Drug uptake | = | 0.54 | % ID/g | ALA2344430 | % ID/g | Rattus norvegicus | |||
8. | ALA2335071 | 1, [18F]4F-MHPG | Drug uptake | = | 0.07 | % ID/g | ALA2344429 | % ID/g | Rattus norvegicus | |||
9. | ALA2335071 | 1, [18F]4F-MHPG | Ratio | = | 1 | ALA2344428 | ||||||
10. | ALA2335071 | 1, [18F]4F-MHPG | Drug uptake | 0 | ALA2344427 | Active | ||||||
11. | ALA2335071 | 1, [18F]4F-MHPG | Drug uptake | 0 | ALA2344425 | Not Active | ||||||
12. | ALA2335071 | 1, [18F]4F-MHPG | Drug uptake | 0 | ALA2344426 | Active | ||||||
13. | ALA2335071 | 1, [18F]4F-MHPG | Drug uptake | 0 | ALA2344424 | Active | ||||||
14. | ALA2335071 | 1, [18F]4F-MHPG | Kup | = | 0.77 | ml/min | ALA2429041 | ml/min | ||||
15. | ALA2335071 | 1, [18F]4F-MHPG | t1/2 | > | 24 | hr | ALA2429040 | hr | ||||
16. | ALA2335071 | 1, [18F]4F-MHPG | Drug uptake | 0 | ALA2429039 | Active | ||||||
17. | ALA2335071 | 1, [18F]4F-MHPG | Drug uptake | 0 | ALA2429038 | Not Active | ||||||
18. | ALA2335071 | 1, [18F]4F-MHPG | Drug uptake | 0 | ALA2429037 | Not Active | ||||||
19. | ALA2335071 | 1, [18F]4F-MHPG | Ratio | = | 3 | ALA2429036 | ||||||
20. | ALA2335071 | 1, [18F]4F-MHPG | Ratio | = | 2.5 | ALA2429035 |