# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2338803 | 30 | IC50 | = | 1.5 | nM | ALA2343135 | 8.82 | nM | Homo sapiens | ||
2. | ALA2338803 | 30 | IC50 | = | 7 | nM | ALA2343132 | 8.15 | nM | Homo sapiens | ||
3. | ALA2338803 | 30 | IC50 | = | 4.4 | nM | ALA2343131 | 8.36 | nM | Mus musculus | ||
4. | ALA2338803 | 30 | IC50 | = | 16 | nM | ALA2343130 | 7.80 | nM | Rattus norvegicus | ||
5. | ALA2338803 | 30 | Drug uptake | = | 460 | ng/ml | ALA2343136 | ng/ml | Mus musculus | |||
6. | ALA2338803 | 30 | Cp | = | 6540 | ng/ml | ALA2343137 | ng/ml | Mus musculus | |||
7. | ALA2338803 | 30 | Activity | 0 | ALA2343129 | Active | Mus musculus | |||||
8. | ALA2338803 | 30 | Activity | 0 | ALA2343138 | Not Active | Mus musculus | |||||
9. | ALA2338803 | 30 | Stability | = | 51 | % | ALA3384566 | % | Rattus norvegicus | |||
10. | ALA2338803 | 30 | Stability | = | 69 | % | ALA3384563 | % | Rattus norvegicus | |||
11. | ALA2338803 | 30 | CL | = | 39 | ml/min.kg | ALA3384569 | mL.min-1.kg-1 | Mus musculus | |||
12. | ALA2338803 | 30 | F | = | 31 | % | ALA3384568 | % | Mus musculus | |||
13. | ALA2338803 | 30 | Stability | = | 62 | % | ALA3384567 | % | Homo sapiens | |||
14. | ALA2338803 | 30 | Stability | = | 59 | % | ALA3384565 | % | ||||
15. | ALA2338803 | 30 | Stability | = | 81 | % | ALA3384564 | % | Homo sapiens | |||
16. | ALA2338803 | 30 | Stability | = | 77 | % | ALA3384562 | % | ||||
17. | ALA2338803 | 30 | IC50 | = | 11 | nM | ALA3888090 | 7.96 | 372199 | nM | Homo sapiens | |
18. | ALA2338803 | 30 | IC50 | = | 7 | nM | ALA3887716 | 8.15 | 349662 | nM | Homo sapiens | |
19. | ALA2338803 | 30 | IC50 | = | 1.5 | nM | ALA3887715 | 8.82 | 349629 | nM | Homo sapiens | |
20. | ALA2338803 | 30 | Stability | = | 59 | % | ALA3788102 | % |