# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2347575 | 3r, diastereomeric mixture | IC50 | = | 13.1 | nM | ALA2349751 | 7.88 | nM | Homo sapiens | ||
2. | ALA2347575 | 3r, diastereomeric mixture | IC50 | = | 3.3 | uM | ALA2349750 | 5.48 | nM | Homo sapiens | ||
3. | ALA2347575 | 3r, diastereomeric mixture | IC50 | = | 2.6 | uM | ALA2349749 | 5.58 | nM | Homo sapiens | ||
4. | ALA2347575 | 3r, diastereomeric mixture | IC50 | = | 2 | uM | ALA2349748 | 5.70 | nM | Homo sapiens | ||
5. | ALA2347575 | 3r, diastereomeric mixture | IC50 | = | 1.6 | uM | ALA2349746 | 5.80 | nM | Homo sapiens | ||
6. | ALA2347575 | 3r, diastereomeric mixture | IC50 | = | 2.3 | uM | ALA2349747 | 5.64 | nM | Homo sapiens | ||
7. | ALA2347575 | 3r, diastereomeric mixture | IC50 | = | 2.7 | uM | ALA2349745 | 5.57 | nM | Homo sapiens | ||
8. | ALA2347575 | 3r, diastereomeric mixture | IC50 | = | 71 | nM | ALA2349744 | 7.15 | nM | Homo sapiens | ||
9. | ALA2347575 | 3r, diastereomeric mixture | IC50 | = | 97 | nM | ALA2349743 | 7.01 | nM | Homo sapiens | ||
10. | ALA2347575 | 3r, diastereomeric mixture | IC50 | = | 165 | nM | ALA2349742 | 6.78 | nM | Homo sapiens | ||
11. | ALA2347575 | 3r, diastereomeric mixture | INH | = | 2.1 | uM | ALA2349741 | uM | Homo sapiens | |||
12. | ALA2347575 | 3r, diastereomeric mixture | Ratio IC50 | > | 13 | ALA2349740 | Homo sapiens | |||||
13. | ALA2347575 | 3r, diastereomeric mixture | Ratio IC50 | > | 9 | ALA2349739 | Homo sapiens | |||||
14. | ALA2347575 | 3r, diastereomeric mixture | Ratio IC50 | > | 9 | ALA2349737 | Homo sapiens | |||||
15. | ALA2347575 | 3r, diastereomeric mixture | Ratio IC50 | > | 9 | ALA2349738 | Homo sapiens | |||||
16. | ALA2347575 | 3r, diastereomeric mixture | Ratio IC50 | > | 9 | ALA2349736 | Homo sapiens | |||||
17. | ALA2347575 | 3r, diastereomeric mixture | Ratio IC50 | > | 9 | ALA2349734 | Homo sapiens | |||||
18. | ALA2347575 | 3r, diastereomeric mixture | Ratio IC50 | > | 9 | ALA2349735 | Homo sapiens | |||||
19. | ALA2347575 | 3r, diastereomeric mixture | Activity | = | 1.5 | % | ALA2349733 | % | Homo sapiens | |||
20. | ALA2347575 | 3r, diastereomeric mixture | Activity | = | 45.6 | % | ALA2349732 | % | Homo sapiens |