# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2348339 | 15k | Activity | = | 28 | % | ALA4388737 | % | Homo sapiens | |||
2. | ALA2348339 | 15k | INH | = | 49 | % | ALA4388746 | % | Homo sapiens | |||
3. | ALA2348339 | 15k | INH | = | 34 | % | ALA4388745 | % | Homo sapiens | |||
4. | ALA2348339 | 15k | INH | = | 96 | % | ALA4388744 | % | Homo sapiens | |||
5. | ALA2348339 | 15k | INH | = | 71 | % | ALA4388743 | % | Homo sapiens | |||
6. | ALA2348339 | 15k | INH | = | 14 | % | ALA4388738 | % | Homo sapiens | |||
7. | ALA2348339 | 15k | F | = | 14 | % | ALA4806861 | % | ||||
8. | ALA2348339 | 15k | AUC | = | 9 | ng.hr/ml | ALA4806860 | ng.hr.mL-1 | ||||
9. | ALA2348339 | 15k | t1/2 | = | 0.86 | hr | ALA4806859 | hr | ||||
10. | ALA2348339 | 15k | Cmax | = | 6.7 | ng/ml | ALA4806858 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
11. | ALA2348339 | 15k | AUC | = | 32 | ng.hr/ml | ALA4806857 | ng.hr.mL-1 | ||||
12. | ALA2348339 | 15k | t1/2 | = | 0.25 | hr | ALA4806856 | hr | ||||
13. | ALA2348339 | 15k | Kel | = | 2.78 | /hr | ALA4806855 | /hr | ||||
14. | ALA2348339 | 15k | Vd | = | 4.23 | L/Kg | ALA4806854 | L.kg-1 | ||||
15. | ALA2348339 | 15k | C0 | = | 118 | ng/ml | ALA4806853 | ng/ml | ||||
16. | ALA2348339 | 15k | EC200 | = | 138.8 | nM | ALA4806369 | nM | Homo sapiens | |||
17. | ALA2348339 | 15k | IC50 | = | 50.6 | nM | ALA4806367 | 7.30 | nM | Homo sapiens | ||
18. | ALA2348339 | 15k | INH | 0 | ALA4742533 | Active | % | Homo sapiens | ||||
19. | ALA2348339 | 15k | INH | 0 | ALA4742532 | Active | % | Homo sapiens | ||||
20. | ALA2348339 | 15k | ECmax | = | 30 | % | ALA4742531 | % | Mus musculus |