# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2349471 | (R)-63 | Fu | 0 | ALA2351998 | Not Determined | Rattus norvegicus | |||||
2. | ALA2349471 | (R)-63 | Fu | = | 0.49 | ALA2351996 | ||||||
3. | ALA2349471 | (R)-63 | Fu | 0 | ALA2351997 | Not Determined | Rattus norvegicus | |||||
4. | ALA2349471 | (R)-63 | Fu | = | 0.1 | ALA2351995 | ||||||
5. | ALA2349471 | (R)-63 | CLH | = | 28 | ml/min.kg | ALA2351994 | mL.min-1.kg-1 | Rattus norvegicus | |||
6. | ALA2349471 | (R)-63 | CLH | = | 12 | ml/min.kg | ALA2351993 | mL.min-1.kg-1 | Cavia porcellus | |||
7. | ALA2349471 | (R)-63 | CLH | = | 29 | ml/min.kg | ALA2351992 | mL.min-1.kg-1 | ||||
8. | ALA2349471 | (R)-63 | CLH | = | 3 | ml/min.kg | ALA2351991 | mL.min-1.kg-1 | Homo sapiens | |||
9. | ALA2349471 | (R)-63 | Cp(f) | = | 3019 | nM | ALA2351975 | nM | ||||
10. | ALA2349471 | (R)-63 | Cp(f) | = | 6673 | nM | ALA2351973 | nM | ||||
11. | ALA2349471 | (R)-63 | Drug uptake | = | 888 | nM | ALA2350193 | nM | ||||
12. | ALA2349471 | (R)-63 | Drug uptake | = | 5609 | nM | ALA2350192 | nM | ||||
13. | ALA2349471 | (R)-63 | Activity | = | 30 | % | ALA2351360 | % | Cavia porcellus | |||
14. | ALA2349471 | (R)-63 | Activity | = | 70 | % | ALA2351099 | % | Cavia porcellus | |||
15. | ALA2349471 | (R)-63 | IC50 | = | 1348 | nM | ALA2352293 | 5.87 | nM | Homo sapiens | ||
16. | ALA2349471 | (R)-63 | IC50 | = | 88464 | nM | ALA2352017 | 4.05 | nM | Homo sapiens | ||
17. | ALA2349471 | (R)-63 | Ratio IC50 | = | 66 | ALA2352016 | ||||||
18. | ALA2349471 | (R)-63 | EC50 | = | 170 | nM | ALA2352015 | 6.77 | nM | Homo sapiens | ||
19. | ALA2349471 | (R)-63 | Ratio | = | 8 | ALA2352014 | Sus scrofa | |||||
20. | ALA2349471 | (R)-63 | Papp | = | 26 | ucm/s | ALA2352013 | ucm/s | Sus scrofa |