# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2375520 | 4, SEP342 | Kd | = | 4.2 | uM | ALA2378321 | 5.38 | nM | Homo sapiens | ||
2. | ALA2375520 | 4, SEP342 | Kd | = | 4.2 | uM | ALA2378322 | 5.38 | nM | Homo sapiens | ||
3. | ALA2375520 | 4, SEP342 | Kd | = | 4 | uM | ALA2378323 | 5.40 | nM | Homo sapiens | ||
4. | ALA2375520 | 4, SEP342 | Kd | = | 3.6 | uM | ALA2378324 | 5.44 | nM | Homo sapiens | ||
5. | ALA2375520 | 4, SEP342 | EC50 | = | 1.5 | uM | ALA2378370 | 5.82 | nM | Rattus norvegicus | ||
6. | ALA2375520 | 4, SEP342 | Drug uptake | < | 1 | uM | ALA2378378 | uM | Mus musculus | |||
7. | ALA2375520 | 4, SEP342 | INH | 0 | ALA2378379 | Active | % | Mus musculus | ||||
8. | ALA2375520 | 4, SEP342 | Ki | = | 1.7 | nM | ALA2378382 | 8.77 | nM | Homo sapiens | ||
9. | ALA2375520 | 4, SEP342 | pIC50 | = | 8.51 | ALA2378383 | 8.51 | nM | Homo sapiens | |||
10. | ALA2375520 | 4, SEP342 | Kd | = | 1.9 | uM | ALA2378384 | 5.72 | nM | Homo sapiens | ||
11. | ALA2375520 | 4, SEP342 | Papp | = | 29 | 10'-6 cm/s | ALA4376726 | 10'-6 cm/s | ||||
12. | ALA2375520 | 4, SEP342 | Ratio | = | 1.2 | ALA4376724 | ||||||
13. | ALA2375520 | 4, SEP342 | Ratio | = | 0.22 | ALA4376723 | ||||||
14. | ALA2375520 | 4, SEP342 | Ratio | = | 10 | ALA4376720 | ||||||
15. | ALA2375520 | 4, SEP342 | K(p,uu,brain) | = | 1.1 | ALA4376721 | ||||||
16. | ALA2375520 | 4, SEP342 | Ratio | = | 9.7 | ALA4376722 | ||||||
17. | ALA2375520 | 4, SEP342 | Ct | = | 17 | ng/ml | ALA4376719 | ng/ml | ||||
18. | ALA2375520 | 4, SEP342 | Ct | = | 4.7 | ng/ml | ALA4376718 | ng/ml | ||||
19. | ALA2375520 | 4, SEP342 | Ct | = | 180 | ng/ml | ALA4376717 | ng/ml | ||||
20. | ALA2375520 | 4, SEP342 | Ct | = | 24 | ng/ml | ALA4376716 | ng/ml |