# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2376321 | (S)-9 | pIC50 | = | 7.6 | ALA2378971 | 7.60 | nM | Homo sapiens | |||
2. | ALA2376321 | (S)-9 | pIC50 | = | 8.2 | ALA2378969 | 8.20 | nM | Mus musculus | |||
3. | ALA2376321 | (S)-9 | pIC50 | = | 7.2 | ALA2378968 | 7.20 | nM | Homo sapiens | |||
4. | ALA2376321 | (S)-9 | pIC50 | = | 6.9 | ALA2378967 | 6.90 | nM | Homo sapiens | |||
5. | ALA2376321 | (S)-9 | pKa | = | 7.9 | ALA2378965 | ||||||
6. | ALA2376321 | (S)-9 | CLH | = | 2.8 | microL/min/mg | ALA2378966 | mL.min-1.g-1 | Homo sapiens | |||
7. | ALA2376321 | (S)-9 | Papp | = | 1.1 | ucm/s | ALA2378964 | ucm/s | Homo sapiens | |||
8. | ALA2376321 | (S)-9 | Ratio | = | 0.5 | ALA2378962 | Homo sapiens | |||||
9. | ALA2376321 | (S)-9 | INH | 0 | ALA2378961 | Not Active | % | |||||
10. | ALA2376321 | (S)-9 | INH | 0 | ALA2378960 | Not Active | % | |||||
11. | ALA2376321 | (S)-9 | Drug metabolism | = | 100 | % | ALA2378959 | % | Homo sapiens | |||
12. | ALA2376321 | (S)-9 | pIC50 | < | 5 | ALA2378958 | nM | Homo sapiens | ||||
13. | ALA2376321 | (S)-9 | pIC50 | < | 5 | ALA2378957 | nM | Homo sapiens | ||||
14. | ALA2376321 | (S)-9 | pIC50 | < | 4 | ALA2378918 | nM | Homo sapiens | ||||
15. | ALA2376321 | (S)-9 | pIC50 | < | 4 | ALA2378804 | nM | Homo sapiens |