| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA2381353 | 14n | IC50 | = | 0.021 | uM | ALA2383097 | 7.68 | nM | Homo sapiens | ||
| 2. | ALA2381353 | 14n | Activity | 0 | ALA2382961 | Active | Homo sapiens | |||||
| 3. | ALA2381353 | 14n | INH | 0 | ALA2382960 | Active | % | Homo sapiens | ||||
| 4. | ALA2381353 | 14n | INH | 0 | ALA2382959 | Not Active | % | Homo sapiens | ||||
| 5. | ALA2381353 | 14n | Activity | 0 | ALA2382958 | Dose-dependent effect | Homo sapiens | |||||
| 6. | ALA2381353 | 14n | INH | 0 | ALA2382957 | Dose-dependent effect | % | Homo sapiens | ||||
| 7. | ALA2381353 | 14n | INH | 0 | ALA2382956 | Dose-dependent effect | % | Homo sapiens | ||||
| 8. | ALA2381353 | 14n | IC50 | = | 3.7 | uM | ALA2382955 | 5.43 | nM | Homo sapiens | ||
| 9. | ALA2381353 | 14n | IC50 | = | 6.9 | uM | ALA2382954 | 5.16 | nM | Homo sapiens | ||
| 10. | ALA2381353 | 14n | Activity | 0 | ALA2382952 | Dose-dependent effect | Homo sapiens | |||||
| 11. | ALA2381353 | 14n | Activity | 0 | ALA2382953 | Active | Homo sapiens | |||||
| 12. | ALA2381353 | 14n | Activity | = | 32 | % | ALA2382951 | % | Homo sapiens | |||
| 13. | ALA2381353 | 14n | Activity | = | 40 | % | ALA2382950 | % | Homo sapiens | |||
| 14. | ALA2381353 | 14n | Cmax | = | 9594 | ug/L | ALA2382949 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
| 15. | ALA2381353 | 14n | Cmax | = | 5115 | ug/L | ALA2382948 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
| 16. | ALA2381353 | 14n | Tmax | = | 0.033 | hr | ALA2382947 | hr | Rattus norvegicus | |||
| 17. | ALA2381353 | 14n | Tmax | = | 1.25 | hr | ALA2382946 | hr | Rattus norvegicus | |||
| 18. | ALA2381353 | 14n | t1/2 | = | 2.1 | hr | ALA2382945 | hr | Rattus norvegicus | |||
| 19. | ALA2381353 | 14n | t1/2 | = | 1.5 | hr | ALA2382943 | hr | Rattus norvegicus | |||
| 20. | ALA2381353 | 14n | AUC | = | 4217 | ug.hr/L | ALA2382944 | ng.hr.mL-1 | Rattus norvegicus |
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