| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA2381936 | 31 | IC50 | = | 3.86 | nM | ALA3888461 | 8.41 | 403134 | nM | Homo sapiens | |
| 2. | ALA2381936 | 31 | IC50 | = | 0.004 | uM | ALA2384487 | 8.40 | nM | Homo sapiens | ||
| 3. | ALA2381936 | 31 | IC50 | > | 85 | uM | ALA2384485 | nM | Homo sapiens | |||
| 4. | ALA2381936 | 31 | EC50 | = | 0.19 | uM | ALA2384483 | 6.72 | nM | Homo sapiens | ||
| 5. | ALA2381936 | 31 | IC50 | = | 0.27 | uM | ALA2384482 | 6.57 | nM | Homo sapiens | ||
| 6. | ALA2381936 | 31 | CLH | = | 51 | microL/min/mg | ALA2384481 | mL.min-1.g-1 | Homo sapiens | |||
| 7. | ALA2381936 | 31 | CLH | = | 87 | microL/min/mg | ALA2384480 | mL.min-1.g-1 | Rattus norvegicus | |||
| 8. | ALA2381936 | 31 | t1/2 | 0 | ALA2384349 | Not Determined | Mus musculus | |||||
| 9. | ALA2381936 | 31 | solubility | = | 94 | ug ml-1 | ALA2384346 | ug.mL-1 | ||||
| 10. | ALA2381936 | 31 | solubility | = | 156 | ug ml-1 | ALA2384347 | ug.mL-1 | ||||
| 11. | ALA2381936 | 31 | solubility | = | 81 | ug ml-1 | ALA2384345 | ug.mL-1 | ||||
| 12. | ALA2381936 | 31 | Papp | 0 | ALA2384344 | Not Determined | Sus scrofa | |||||
| 13. | ALA2381936 | 31 | Ratio | 0 | ALA2384343 | Not Determined | Sus scrofa | |||||
| 14. | ALA2381936 | 31 | IC50 | > | 170 | uM | ALA2384484 | nM | Homo sapiens | |||
| 15. | ALA2381936 | 31 | AUCt | = | 2.24 | uM.hr | ALA2384339 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Mus musculus | ||
| 16. | ALA2381936 | 31 | Cmax | = | 1.3 | uM | ALA2384340 | nM | Mus musculus | |||
| 17. | ALA2381936 | 31 | EC50 | = | 0.19 | uM | ALA2384334 | 6.72 | nM | Homo sapiens | ||
| 18. | ALA2381936 | 31 | IC50 | > | 27 | uM | ALA2384333 | nM | Homo sapiens | |||
| 19. | ALA2381936 | 31 | Activity | = | 3 | % | ALA2384332 | % | Rattus norvegicus | |||
| 20. | ALA2381936 | 31 | Ratio | = | 0.57 | ALA2384331 |
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