# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2386492 | 7b, diastereomer | EC50 | = | 0.6 | uM | ALA2388104 | 6.22 | nM | Homo sapiens | ||
2. | ALA2386492 | 7b, diastereomer | EC50 | = | 1 | uM | ALA2390599 | 6.00 | nM | Homo sapiens | ||
3. | ALA2386492 | 7b, diastereomer | Ratio EC50 | <= | 530 | ALA2390598 | ||||||
4. | ALA2386492 | 7b, diastereomer | IC50 | = | 120 | uM | ALA2390597 | nM | ||||
5. | ALA2386492 | 7b, diastereomer | IC50 | = | 39 | uM | ALA2390596 | 4.41 | nM | |||
6. | ALA2386492 | 7b, diastereomer | IC50 | = | 0.2 | uM | ALA2390594 | 6.70 | nM | Rattus norvegicus | ||
7. | ALA2386492 | 7b, diastereomer | Drug metabolism | = | 2.5 | % | ALA2390592 | % | Homo sapiens | |||
8. | ALA2386492 | 7b, diastereomer | Drug metabolism | = | 2.9 | % | ALA2390591 | % | Homo sapiens | |||
9. | ALA2386492 | 7b, diastereomer | Drug metabolism | 0 | ALA2390590 | Not Determined | Homo sapiens | |||||
10. | ALA2386492 | 7b, diastereomer | Drug metabolism | = | 46 | % | ALA2390589 | % | Homo sapiens | |||
11. | ALA2386492 | 7b, diastereomer | Drug metabolism | 0 | ALA2390588 | Not Determined | Homo sapiens | |||||
12. | ALA2386492 | 7b, diastereomer | Drug metabolism | 0 | ALA2390587 | Not Determined | Homo sapiens | |||||
13. | ALA2386492 | 7b, diastereomer | EC50 | = | 0.4 | uM | ALA2390584 | 6.40 | nM |