| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA2397488 | 7b, diastereomer | Ki | = | 50.5 | nM | ALA2400839 | 7.30 | nM | Rattus norvegicus | ||
| 2. | ALA2397488 | 7b, diastereomer | CLH | = | 16 | microL/min/mg | ALA2400838 | mL.min-1.g-1 | Homo sapiens | |||
| 3. | ALA2397488 | 7b, diastereomer | t1/2 | = | 103 | min | ALA2400836 | hr | Homo sapiens | |||
| 4. | ALA2397488 | 7b, diastereomer | Drug uptake | = | 14.9 | pmol/min | ALA2400834 | pmol/min | Cricetulus griseus | |||
| 5. | ALA2397488 | 7b, diastereomer | Drug uptake | = | 10.9 | pmol/min | ALA2400835 | pmol/min | Cricetulus griseus | |||
| 6. | ALA2397488 | 7b, diastereomer | Ratio | = | 1.4 | ALA2400833 | ||||||
| 7. | ALA2397488 | 7b, diastereomer | Papp | = | 0.76 | ucm/s | ALA2400832 | ucm/s | Homo sapiens | |||
| 8. | ALA2397488 | 7b, diastereomer | Papp | = | 76.2 | ucm/s | ALA2400831 | ucm/s | Homo sapiens | |||
| 9. | ALA2397488 | 7b, diastereomer | Ratio | = | 95 | ALA2400830 | Homo sapiens |
The page will load shortly, Thanks for your patience!