# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2398729 | 51, diastereomeric mixture | IC50 | = | 0.8 | nM | ALA2399021 | 9.10 | nM | Homo sapiens | ||
2. | ALA2398729 | 51, diastereomeric mixture | IC50 | = | 2.9 | nM | ALA2398869 | 8.54 | nM | Homo sapiens | ||
3. | ALA2398729 | 51, diastereomeric mixture | EC60 | > | 50 | uM | ALA2398843 | uM | Homo sapiens | |||
4. | ALA2398729 | 51, diastereomeric mixture | EC20 | = | 5.3 | uM | ALA2398843 | uM | Homo sapiens | |||
5. | ALA2398729 | 51, diastereomeric mixture | Stability | = | 43 | % | ALA2398841 | % | Homo sapiens | |||
6. | ALA2398729 | 51, diastereomeric mixture | Stability | = | 75 | % | ALA2398839 | % | Rattus norvegicus | |||
7. | ALA2398729 | 51, diastereomeric mixture | Stability | = | 60 | % | ALA2398840 | % | Mus musculus | |||
8. | ALA2398729 | 51, diastereomeric mixture | Stability | = | 22 | % | ALA2398837 | % | ||||
9. | ALA2398729 | 51, diastereomeric mixture | INH | = | 5 | % | ALA2398838 | % | ||||
10. | ALA2398729 | 51, diastereomeric mixture | INH | = | -4 | % | ALA2398836 | % |