# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2398747 | 27 | Ki | = | 0.7 | nM | ALA3706150 | 9.15 | 235353 | nM | Homo sapiens | |
2. | ALA2398747 | 27 | IC50 | = | 1.4 | nM | ALA2399021 | 8.85 | nM | Homo sapiens | ||
3. | ALA2398747 | 27 | IC50 | = | 2.5 | nM | ALA2398869 | 8.60 | nM | Homo sapiens | ||
4. | ALA2398747 | 27 | EC20 | = | 0.4 | uM | ALA2398843 | uM | Homo sapiens | |||
5. | ALA2398747 | 27 | EC60 | = | 1.4 | uM | ALA2398843 | uM | Homo sapiens | |||
6. | ALA2398747 | 27 | Stability | = | 47 | % | ALA2398841 | % | Homo sapiens | |||
7. | ALA2398747 | 27 | Stability | = | 50 | % | ALA2398839 | % | Rattus norvegicus | |||
8. | ALA2398747 | 27 | Stability | = | 26 | % | ALA2398840 | % | Mus musculus | |||
9. | ALA2398747 | 27 | Stability | = | 4 | % | ALA2398837 | % | ||||
10. | ALA2398747 | 27 | INH | = | 52 | % | ALA2398838 | % | ||||
11. | ALA2398747 | 27 | INH | = | 50 | % | ALA2398836 | % |