# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2403843 | 18a | IC50 | = | 1.1 | uM | ALA2406355 | 5.96 | nM | Homo sapiens | ||
2. | ALA2403843 | 18a | CLH | = | 8 | microL/min/mg | ALA2406358 | mL.min-1.g-1 | Homo sapiens | |||
3. | ALA2403843 | 18a | INH | = | 9.8 | uM | ALA2406357 | uM | Homo sapiens | |||
4. | ALA2403843 | 18a | CLH | = | 14 | microL/min/mg | ALA2406360 | mL.min-1.g-1 | Rattus norvegicus | |||
5. | ALA2403843 | 18a | IC50 | = | 14.6 | nM | ALA2406365 | 7.84 | nM | Homo sapiens | ||
6. | ALA2403843 | 18a | CLH | = | 15 | microL/min/mg | ALA2406359 | mL.min-1.g-1 | Mus musculus | |||
7. | ALA2403843 | 18a | IC50 | = | 15.6 | nM | ALA2406362 | 7.81 | nM | Homo sapiens | ||
8. | ALA2403843 | 18a | IC50 | = | 20 | uM | ALA2406353 | 4.70 | nM | Homo sapiens | ||
9. | ALA2403843 | 18a | solubility | = | 144 | uM | ALA2406356 | nM | ||||
10. | ALA2403843 | 18a | IC50 | = | 375.3 | nM | ALA2406363 | 6.43 | nM | Homo sapiens | ||
11. | ALA2403843 | 18a | IC50 | = | 4077 | nM | ALA2406364 | 5.39 | nM | Mus musculus | ||
12. | ALA2403843 | 18a | Drug metabolism | < | 1 | % | ALA2406361 | % | Homo sapiens |