# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2407295 | 17 | K | > | 100 | uM | ALA3413044 | uM | Homo sapiens | |||
2. | ALA2407295 | 17 | Activity | = | 1.9 | % | ALA3413043 | % | Mus musculus | |||
3. | ALA2407295 | 17 | INH | = | 5.2 | % | ALA3413041 | % | ||||
4. | ALA2407295 | 17 | IC50 | = | 0.74 | uM | ALA3413040 | 6.13 | nM | |||
5. | ALA2407295 | 17 | INH | = | 1.9 | % | ALA3413038 | % | ||||
6. | ALA2407295 | 17 | INH | 0 | ALA3413040 | Dose-dependent effect | % | |||||
7. | ALA2407295 | 17 | INH | 0 | ALA3413041 | Dose-dependent effect | % | |||||
8. | ALA2407295 | 17 | INH | = | 22.2 | % | ALA3413039 | % | Mus musculus | |||
9. | ALA2407295 | 17 | Kinetic_solubility | = | 6.7 | 10'-4mg/ml | ALA4384339 | 10'-4mg/ml | ||||
10. | ALA2407295 | 17 | Kinetic_solubility | = | 1.6 | 10'-4mg/ml | ALA4384338 | 10'-4mg/ml | ||||
11. | ALA2407295 | 17 | CLH | < | 3 | ml/min | ALA4384337 | ml/min | ||||
12. | ALA2407295 | 17 | t1/2 | > | 231 | min | ALA4384336 | hr | ||||
13. | ALA2407295 | 17 | GI50 | > | 10 | uM | ALA4384335 | nM | ||||
14. | ALA2407295 | 17 | Activity | 0 | ALA3271533 | Not Active | Mus musculus | |||||
15. | ALA2407295 | 17 | Activity | 0 | ALA3271531 | Active | Mus musculus | |||||
16. | ALA2407295 | 17 | INH | 0 | ALA3271524 | Not Active | % | |||||
17. | ALA2407295 | 17 | Activity | 0 | ALA3271523 | Not Active | ||||||
18. | ALA2407295 | 17 | INH | 0 | ALA3271522 | Not Active | % | |||||
19. | ALA2407295 | 17 | Activity | 0 | ALA3271521 | Not Active | ||||||
20. | ALA2407295 | 17 | INH | 0 | ALA3271520 | Active | % |