# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2407897 | 47 | IC50 | = | 2 | nM | ALA2410318 | 8.70 | nM | Homo sapiens | ||
2. | ALA2407897 | 47 | IC50 | > | 10 | uM | ALA2410316 | nM | Homo sapiens | |||
3. | ALA2407897 | 47 | IC50 | > | 10 | uM | ALA2410317 | nM | Homo sapiens | |||
4. | ALA2407897 | 47 | IC50 | > | 10 | uM | ALA2410315 | nM | Homo sapiens | |||
5. | ALA2407897 | 47 | GI50 | = | 0.01 | uM | ALA2410313 | nM | Homo sapiens | |||
6. | ALA2407897 | 47 | GI50 | = | 0.01 | uM | ALA2410312 | nM | Homo sapiens | |||
7. | ALA2407897 | 47 | GI50 | = | 0.002 | uM | ALA2410310 | nM | Homo sapiens | |||
8. | ALA2407897 | 47 | GI50 | = | 1.9 | uM | ALA2410311 | nM | Homo sapiens | |||
9. | ALA2407897 | 47 | GI50 | = | 0.48 | uM | ALA2410309 | nM | Homo sapiens | |||
10. | ALA2407897 | 47 | IC50 | = | 10 | uM | ALA2410121 | 5.00 | nM | Homo sapiens | ||
11. | ALA2407897 | 47 | IC50 | > | 10 | uM | ALA2410119 | nM | Homo sapiens | |||
12. | ALA2407897 | 47 | IC50 | = | 9 | uM | ALA2410120 | 5.05 | nM | Homo sapiens | ||
13. | ALA2407897 | 47 | IC50 | = | 1 | uM | ALA2410118 | 6.00 | nM | Homo sapiens | ||
14. | ALA2407897 | 47 | IC50 | = | 1.3 | uM | ALA2410117 | 5.89 | nM | Homo sapiens | ||
15. | ALA2407897 | 47 | permeability | = | 276 | ucm/s | ALA2410116 | ucm/s | ||||
16. | ALA2407897 | 47 | IC50 | = | 4 | nM | ALA3420030 | 8.40 | nM | Homo sapiens | ||
17. | ALA2407897 | 47 | AUC | = | 0.83 | ug.hr/ml | ALA3364625 | ng.hr.mL-1 | Mus musculus | |||
18. | ALA2407897 | 47 | Cmax | = | 0.87 | ug ml-1 | ALA3364624 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Mus musculus | ||
19. | ALA2407897 | 47 | t1/2 | = | 40 | min | ALA3364623 | hr | Homo sapiens | |||
20. | ALA2407897 | 47 | t1/2 | = | 7 | min | ALA3364622 | hr | Mus musculus |